Powder: -20°C for 3 years | In solvent: -80°C for 1 year
5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 273,500 |
5 mg | 在庫あり | ¥ 548,500 |
10 mg | 在庫あり | ¥ 739,000 |
25 mg | 在庫あり | ¥ 1,099,500 |
50 mg | 在庫あり | ¥ 1,482,500 |
100 mg | 在庫あり | ¥ 2,001,500 |
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 649,500 |
説明 | 5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity. |
In vitro | 5-HT2 antagonist 1 displays dose-dependent inhibition of serotonin (erotonin)-induced contraction in guinea pig mesenteric artery, exhibiting 45%, 88%, and 93% inhibition at concentrations of 10 nM, 100 nM, and 1000 nM, respectively. Conversely, it demonstrates minimal inhibition of norepinephrine-induced contraction in guinea pig aorta, with 1% and 10% inhibition at 10 nM and 100 nM, respectively[1]. |
分子量 | 400.49 |
分子式 | C22H29FN4O2 |
CAS No. | 191592-09-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 45 mg/mL (112.36 mM)
You can also refer to dose conversion for different animals. 詳細
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5-HT2 antagonist 1 191592-09-3 GPCR/G Protein Neuroscience 5-HT Receptor 5HT2 antagonist 1 5 HT2 antagonist 1 5-HT-2 antagonist 1 Inhibitor inhibitor inhibit