Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Anxiolytic/nonsedative agent-1 (TCS 1205) is a potent and selective GABAA agonist. Anxiolytic/nonsedative agent-1 shows appreciable affinity for the BzR in bovine brain membranes with Kis of 14, 121, 239 nM for α1β2γ2, α2β2γ2, α5β3γ2, respectively. Anxiolytic/nonsedative agent-1 shows α2 selective efficacy in vitro and anxioselective effects in vivo.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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1 mg | 在庫あり | ¥ 22,500 | |||
2 mg | 在庫あり | ¥ 34,000 | |||
5 mg | 在庫あり | ¥ 45,000 | |||
10 mg | 在庫あり | ¥ 59,000 | |||
25 mg | 在庫あり | ¥ 133,500 | |||
50 mg | 在庫あり | ¥ 190,500 | |||
100 mg | 在庫あり | ¥ 264,000 | |||
500 mg | 在庫あり | ¥ 523,500 |
説明 | Anxiolytic/nonsedative agent-1 (TCS 1205) is a potent and selective GABAA agonist. Anxiolytic/nonsedative agent-1 shows appreciable affinity for the BzR in bovine brain membranes with Kis of 14, 121, 239 nM for α1β2γ2, α2β2γ2, α5β3γ2, respectively. Anxiolytic/nonsedative agent-1 shows α2 selective efficacy in vitro and anxioselective effects in vivo. |
別名 | TCS 1205 |
分子量 | 337.33 |
分子式 | C18H15N3O4 |
CAS No. | 355022-97-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 1mg/ml, Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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Anxiolytic/nonsedative agent-1 355022-97-8 Membrane transporter/Ion channel Neuroscience GABA Receptor TCS-1205 TCS1205 TCS 1205 Inhibitor inhibitor inhibit