Powder: -20°C for 3 years | In solvent: -80°C for 1 year
BJJF078, an aminopiperidine derivative, is a potent inhibitor of recombinant human and mouse glutamine aminotransferase (TG2) activity, with IC50 values of 41 and 54 nM for human and mouse glutamine aminotransferase, respectively.BJJF078 inhibits TG1 enzyme, with an IC50 of 0.16 μM.BJJF078 can be used to study multiple sclerosis (MS). BJJF078 can be used to study multiple sclerosis (MS).
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 12,500 | |||
5 mg | 在庫あり | ¥ 25,500 | |||
10 mg | 在庫あり | ¥ 36,500 | |||
25 mg | 在庫あり | ¥ 61,000 | |||
50 mg | 在庫あり | ¥ 91,000 | |||
100 mg | 在庫あり | ¥ 135,500 |
説明 | BJJF078, an aminopiperidine derivative, is a potent inhibitor of recombinant human and mouse glutamine aminotransferase (TG2) activity, with IC50 values of 41 and 54 nM for human and mouse glutamine aminotransferase, respectively.BJJF078 inhibits TG1 enzyme, with an IC50 of 0.16 μM.BJJF078 can be used to study multiple sclerosis (MS). BJJF078 can be used to study multiple sclerosis (MS). |
ターゲット&IC50 | TGase 1:0.16 μM, TG2 (human):41 nM, TG2 (mouse):54 nM |
分子量 | 523.6 |
分子式 | C27H29N3O6S |
CAS No. | 2531244-56-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 60 mg/mL (114.59 mM)
You can also refer to dose conversion for different animals. 詳細
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BJJF078 2531244-56-9 Proteases/Proteasome Glutaminase BJJF 078 BJJF-078 Inhibitor inhibitor inhibit