Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CYP1B1-IN-5 is a selective and potent cytochrome P450 1B1 (CYP1B1) inhibitor with an IC50 of 4.7 nM.CYP1B1-IN-5 can be used for the study of metabolism-related diseases.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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1 mg | 在庫あり | ¥ 45,000 | |||
5 mg | 在庫あり | ¥ 111,000 | |||
10 mg | 在庫あり | ¥ 159,000 | |||
25 mg | 在庫あり | ¥ 248,000 | |||
50 mg | 在庫あり | ¥ 342,000 | |||
100 mg | 在庫あり | ¥ 452,500 | |||
500 mg | 在庫あり | ¥ 902,000 |
説明 | CYP1B1-IN-5 is a selective and potent cytochrome P450 1B1 (CYP1B1) inhibitor with an IC50 of 4.7 nM.CYP1B1-IN-5 can be used for the study of metabolism-related diseases. |
ターゲット&IC50 | CYP1A1:190.7 nM, CYP1B1:4.7 nM, CYP1A2:585.7 nM |
In vitro | CYP1B1-IN-5 (Compound 6q) binds to the binding pocket of CYP1B1 by forming π-π stacking interactions with residues Phe231, Phe134 and heme.[1] |
分子量 | 349.12 |
分子式 | C14H8INO2 |
CAS No. | 176442-56-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 5.63 mg/mL (16.11 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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CYP1B1-IN-5 176442-56-1 Metabolism P450 Inhibitor inhibitor inhibit