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TP1073 |
Neuropeptide W-23(human)
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NPW-23 |
Others
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Neuropeptide W-23(human) (NPW-23) is an endogenous ligand for NPBW1 and NPBW2. |
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T62656 |
GPR81 agonist 1
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GPR
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GPR81 agonist 1 is a potent and selective GPR81 agonist with high affinity for human and mouse GPR81.GPR81 agonist 1 inhibits lipolysis of differentiated 3T3-L1 adipocytes, improves insulin sensitivity and glycaemic cont... |
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T62261 |
GPR84 antagonist 1
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GPR84 antagonist 1 is a highly selective, high-affinity competitive antagonist of human GPR84. |
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T72536 |
GPR84 antagonist 2
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GPR84 Antagonist 2, a potent and selective GPR84 antagonist (IC 50 = 8.95 nM), demonstrates oral activity and significantly enhances potency in calcium mobilization assays. It effectively inhibits neutrophil and macropha... |
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T11462 |
GPR84 antagonist 8
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GPR
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T79902 |
GPR88 agonist 2
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GPR88 agonist 2 (compound 53) serves as a potent, brain-penetrant agonist of GPR88, exhibiting an EC50 of 14 µM in the GPR88 cAMP functional assay [1]. |
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T79901 |
GPR88-IN-1
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GPR88-IN-1 is a GPR88 antagonist that may be utilized for the study of central nervous system disorders [1]. |
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T72772 |
GPR81 agonist 2
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GPR81 agonist 2 is a potent agonist targeting the GPR81 receptor, demonstrating EC50 values of 0.023 µM for hGPR81 and 0.123 µM for hGPR109A, respectively. |
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T62918 |
GPR84 antagonist 3
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GPR84 Antagonist 3 (compound 42), a potent inhibitor of the G-protein-coupled receptor 84 (GPR84), exhibits a pIC50 value of 8.28, indicating strong antagonistic activity by inhibiting GTPγS. Additionally, it possesses a... |
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T81680 |
Neuropeptide W-23 (human) (TFA)
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NPW-23 TFA |
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Neuropeptide W-23 (human) (NPW-23) TFA, representing the active form of Neuropeptide W, functions as an endogenous agonist for both NPBW1 (GPR7) and NPBW2 (GPR8) receptors [1]. |
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T82862 |
Biotinyl-neuropeptide W-23 (human)
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Biotinyl-neuropeptide W-23 (human) is a biotinylated form of neuropeptide W-23 (human), which functions as an agonist for the NPBW1 (GPR7) and NPBW2 (GPR8) receptors [1] [2]. |
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T83547 |
(Des-Bromo)-Neuropeptide B (1-23) (human)
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'(Des-Bromo)-Neuropeptide B (1-23) (human)' is an agonist for orphan G-protein-coupled receptors, exhibiting a K i of 1.2 nM for GPR7 (NPBW1) and 341 nM for GPR8 (NPBW2) respectively [1]. |
