ペプチド
抗体
色素試薬
PROTAC
バーチャルスクリーニング
TargetMolキット
Cell Counting Kit-8 (CCK-8)
Inhibitor Cocktails
天然化合物
フェノール類
アルカロイド類
フラボノイド類
阻害剤
血管新生
アポトーシス
オートファジー
細胞周期・チェックポイント
クロマチン・エピジェネティック
細胞骨格シグナル
DNA損傷・DNA修復
内分泌・ホルモン
GPCR/Gタンパク質
免疫・炎症
JAK・STATシグナル
| Cat. No. | 製品名 | CAS No. | Purity | Chemical Structure |
|---|---|---|---|---|
| T3965 | Fevipiprant | 872365-14-5 | 98% |
|
| Fevipiprant is a selective, potent, reversible competitive CRTh2 antagonist. | ||||
| T22986 | MK 1903 | 1268882-43-4 | 98% |
|
| MK 1903 is a potent and selective complete agonist for the hydroxy-carboxylic acid receptor 2 (HCA2). HCA2 is also known as G protein-coupled receptor 109A(GPR10... | ||||
| T4566 | Lodoxamide | 53882-12-5 | 98% |
|
| Lodoxamide is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis. | ||||
| TN1849 | Kuwanon H | 76472-87-2 | 98% |
|
| Kuwanon H, and possibly kuwanon G also, are specific antagonists for the gastrin-releasing peptide (GRP) -preferring receptor and can be useful for studying the ... | ||||
| T12216 | NF-56-EJ40 | 2380230-73-7 | 98% |
|
| NF-56-EJ40 is an effective and highly selective antagonist of human SUCNR1 with an IC50 of 25 nM and a Ki of 33 nM. | ||||
| TP1345 | Kisspeptin-10, human (TFA)(374675-21-5,FREE) | TP1345 | 98% |
|
| Kisspeptin-10, human TFA is a potent vasoconstrictor and angiogenesis inhibitor. Kisspeptin-10, human TFA acts as a tumor metastasis suppressor via its receptor ... | ||||
| T77601 | (2-{[2-(2-fluorophenoxy)ethyl]sulfanyl}-1H-benzimidazol-1-yl)acetic acid | 303134-93-2 | 98% |
|
| (2-{[2-(2-fluorophenoxy)ethyl]sulfanyl}-1H-benzimidazol-1-yl)acetic acid is a prostaglandin-like CRTH2 antagonist with an IC50 < 10 μM, which can be used in stud... | ||||
| T1286 | Vincamine | 1617-90-9 | 98% |
|
| Vincamine is a major alkaloid of Vinca minor L., Apocynaceae. It has been used therapeutically as a vasodilator and antihypertensive agent, particularly in cereb... | ||||
| T1781 | GW9508 | 885101-89-3 | 98% |
|
| GW9508 is a potent and selective agonist for FFA1 (GPR40), stimulates insulin secretion in a glucose-sensitive manner. | ||||
| T2351 | Fasiglifam | 1000413-72-8 | 98% |
|
| TAK875 is a potent, selective and orally bioavailable GPR40 agonist. | ||||
| T2528 | Latanoprost | 130209-82-4 | 98% |
|
| Latanoprost is a prostaglandin F2alpha analogue and a prostanoid selective FP receptor agonist with an ocular hypertensive effect. | ||||
| T36818 | Questiomycin A | 1916-59-2 | 98% |
|
| Questiomycin A is an antibiotic produced in crème fraiche with antibacterial and anticancer activities. Questiomycin A suppresses expression of GRP78, a cell-pro... | ||||
| T12095 | Monomethyl fumarate | 2756-87-8 | 98% |
|
| Monomethyl fumarate is a potent agonist of GPR109A . | ||||
| T15413 | GPR120 Agonist 3 | 1599477-75-4 | 98% |
|
| GPR120-IN-1 is a selective agonist of Gpr120 (logEC50: −7.62). | ||||
| TP1928L1 | [Orn5]-URP acetate | TP1928L1 | 98% |
|
| [Orn5]-URP acetate is an effective and selective Urotensin-II receptor (UT) antagonist (pEC50 = 7.24). [Orn5]-URP exhibits no agonist activity. | ||||
| T4312 | GPR120 Agonist 2 | 1234844-11-1 | 98% |
|
| A potent and selective GPR120 receptor agonist. | ||||
| TN1560 | Dehydroeffusol | 137319-34-7 | 98% |
|
| Dehydroeffusol possesses anti-cancer, anxiolytic and sedative properties, it may antagonize the spasmogenic activity of various agents, and therefore, could be a... | ||||
| T60074 | WAY-622024 | 291528-35-3 | 98% |
|
| WAY-622024 is an agonist of the orphan human GPCR GPR109B. | ||||
| T21622 | Tyrphostin A25 | 118409-58-8 | 98% |
|
| Tyrphostin A25 is a specific EGFR tyrosine kinase inhibitor and GPR35 agonist with an IC50 value of 0.94 μM for GPR35 and an EC50 value of 5.3 μM for GPR35. | ||||
| T9719 | 3-Hydroxyoctanoic Acid | 14292-27-4 | 98% |
|
| 3-Hydroxyoctanoic Acid is one of the hydroxy-carboxylic acids (HCAs) that serve as intermediates of energy metabolism. It is an agonist of the orphan receptor GP... | ||||
