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Search Results for " Thelin "

ターゲット

阻害剤

リコンビナントタンパク質

カタログ番号	製品名	別名	ターゲット
T6672	Sitaxsentan sodium	TBC11251 sodium salt,TBC11251,Thelin,Sitaxentan sodium	Endothelin Receptor
	Sitaxsentan sodium (TBC11251 sodium salt) is a highly selective antagonist of endothelin A receptors.		Endothelin Receptor
T22540L	Ac-Endothelin-1 (16-21), human acetate		Others
	Ac-Endothelin-1 (16-21), human acetate, the principal peptide of the endothelin family, has been shown to have a variety of biological activities in both vascular and nonvascular tissues. The C-terminal fragment, which i...		Others
TP1174	Endothelin-2 (49-69), human	Human endothelin-2,Endothelin-2, human,Endothelin-2 (human, canine)	Others
	Endothelin-2 (49-69), human (Human endothelin-2) is a 21-amino acid vasoactive peptide that binds to G-protein-linked transmembrane receptors, ET-RA and ET-RB.		Others
T19309L1	Endothelin 1 (swine, human) acetate	Endothelin 1 (swine, human) acetate(117399-94-7 free base)	Endothelin Receptor
	Endothelin 1 (swine, human) acetate is a synthetic peptide with the sequence of human and swine Endothelin 1. Endothelin 1 is a potent endogenous vasoconstrictor and acts through two types of receptors ETA and ETB.		Endothelin Receptor
T1006	Propantheline bromide	Neopepulsan,Pro-Banthine,Neometantyl	AChR
	Propantheline bromide (Pro-Banthine) competitively antagonizes acetylcholine activity mediated by muscarinic receptors at neuroeffector sites on smooth muscle and exocrine gland cells. Propantheline Bromide is the bromid...		AChR
TP2143	Endothelin-2 (49-69), human TFA	Endothelin-2 (49-69) (human, canine) TFA,Human endothelin-2 TFA	Others
	Endothelin-2 (49-69), human (TFA) is a 21-amino acid vasoactive peptide that binds to ET-RA and ET-RB.		Others
T82886	Big endothelin-1 (rat 1-39)
	Big endothelin-1 (rat 1-39), a 39-residue peptide, induces a diuretic and natriuretic response in conscious Sprague-Dawley rats and elevates blood pressure in mice [1].
TP2099	[Ala1,3,11,15]-Endothelin
	Selective ETB endothelin receptor agonist (IC50 values are 0.33 and 2200 nM for displacing [125I]-ET-1 from ETB and ETA receptors respectively).
TP1512	[Ala1,3,11,15]-Endothelin TFA
	[Ala1,3,11,15]-Endothelin (TFA) is a highly selective for endothelin A (ETA) and endothelin B (ETB) receptor.[Ala1,3,11,15]-Endothelin is a selective ETB endothelin receptor agonist (IC50 values are 0.33 and 2200 nM for ...
TP1173	Endothelin 3 (Rat,Human) (TFA)	Endothelin-3, human, mouse, rabbit, rat TFA
	Endothelin-3, human, mouse, rabbit, rat TFA is a 21-amino acid vasoactive peptide that specifically interacts with G-protein-linked transmembrane receptors, ET-RA and ET-RB.
T75772	[Ala1,3,11,15]-Endothelin (53-63) (TFA)
	[Ala1,3,11,15]-Endothelin (53-63) (TFA) is a selective ET B agonist with IC50 values ranging from 0.33 nM to 0.61 nM, demonstrating its preference for ET B receptors. It is utilized in the study of vasoconstriction.
T36479	Big Endothelin-1 (1-38), human
	Human Big ET-1 comprises residues 53-90 of the endothelin precursor (preproendothelin). Compared to the mature endothelin-1 (hET-1), the peptide show less vasoconstrictor activity in vitro, but similar pressor effects in...
TP2246	Endothelin-1 (1-15), amide, human		Others
	Endothelin-1 is one of the there isoforms of endothelin (identified as ET-1, -2, -3) with varying regions of expression and binding to at least four known endothelin receptors, ETA, ETB1, ETB2 and ETC.		Others
T19309	Endothelin 1 (swine, human)		Others
	Endothelin 1 (swine, human), a synthetic peptide mirroring the sequence of both human and swine Endothelin 1, functions as a robust endogenous vasoconstrictor by interacting with two receptor types, ETA and ETB.		Others
T75731	Endothelin 1 (swine, human) (TFA)
	Endothelin 1 (swine, human) (TFA) is a synthetic peptide mirroring the sequence of the potent endogenous vasoconstrictor found in both human and swine Endothelin 1. It operates via two receptor types, ET A and ET B [1].
T76564	Endothelin-1 (1-31) (Human)
	Endothelin-1 (1-31) (Human) is a powerful vasoconstrictor and agent for inducing hypertension, originating from the specific hydrolysis of big ET-1 by chymase [1].
T76081	Endothelin 1 (swine, human), Alexa Fluor 488-labeled
	Endothelin 1 (swine, human), Alexa Fluor 488-labeled, is a synthetic peptide corresponding to the sequence of human and swine Endothelin 1, a powerful endogenous vasoconstrictor, and is tagged with Alexa Fluor 488 for fl...
T76564L	Endothelin-1 (1-31) (Human) acetate
	Endothelin-1 (1-31) (Human) acetate, a potent vasoconstrictor and hypertensive agent, is produced through the selective hydrolysis of big ET-1 by chymase [1].
T61453	Propantheline
	Propantheline is an orally active antagonist of muscarinic acetylcholine receptors (mAChRs), commonly employed to investigate smooth muscle dysfunction, hyperhidrosis, smooth muscle spasms or cramps in the stomach, intes...
T22540	Ac-Endothelin-1 (16-21), human		Others
	ENDOTHELIN-1 (ET-1), the principal peptide of the endothelin family, has been shown to have a variety of biological activities in both vascular and nonvascular tissues. The C-terminal fragment, which is a highly cons...		Others
TP1175	Endothelin-3, human, mouse, rabbit, rat	Endothelin 3 (Rat,Human)
	Endothelin-3, human, mouse, rabbit, rat , is a cyclic 21 amino acid peptide. It is an endogenous neuropeptide and potent vasoconstrictor.
T36480	Big Endothelin-1 (1-39), porcine
	The big endothelins comprise residues 53-90 (human big ET-1) and 53-91 (porcine big ET-1) of the endothelin precursor (preproendothelin). Compared to the mature endothelin-1 (ET-1), both peptides show less vasoconstricto...
T78063	Endothelin-1 (1-31) (Human) TFA		ERK
	Endothelin-1 (1-31) (Human) TFA, a potent vasoconstrictor and hypertensive agent, originates from the chymase-mediated selective hydrolysis of big ET-1 [1].		ERK
T76329	[Asn18] Endothelin-1, human
	[Asn18] Endothelin-1, human, a peptide, represents a predominant isoform of Endothelin, significantly contributing to the regulation of vascular function [1].
T33314	Methantheline Bromide	Frenogastrico,Dixamone bromide,Banthine,Asabaine,Methanthelinium bromide
	Methantheline Bromide is a synthetic spasmolytic used to relieve cramps or spasms of the stomach, bowel, and bladder. It is also useful for intestinal or gastric ulcers (peptic ulcer disease), intestinal problems, pancre...
T76305	[Ala2] Endothelin-3, human
	[Ala2] Endothelin-3, human is a linear analog of endothelin-3 (ET-3), characterized by the substitution of Ala for Cys residues. ET-3, a vasoactive peptide produced by human rhabdomyosarcoma cell lines but not expressed ...

Compounds

Sitaxsentan sodium

T6672

Synonym: TBC11251 sodium salt,TBC11251,Thelin,Sitaxentan sodium

Target: Endothelin Receptor

Ac-Endothelin-1 (16-21), human acetate

T22540L

Synonym:

Target: Others

Endothelin-2 (49-69), human

TP1174

Synonym: Human endothelin-2,Endothelin-2, human,Endothelin-2 (human, canine)

Target: Others

Endothelin 1 (swine, human) acetate

T19309L1

Synonym: Endothelin 1 (swine, human) acetate(117399-94-7 free base)

Target: Endothelin Receptor

Propantheline bromide

T1006

Synonym: Neopepulsan,Pro-Banthine,Neometantyl

Target: AChR

Endothelin-2 (49-69), human TFA

TP2143

Synonym: Endothelin-2 (49-69) (human, canine) TFA,Human endothelin-2 TFA

Target: Others

Big endothelin-1 (rat 1-39)

T82886

Synonym:

Target:

[Ala1,3,11,15]-Endothelin

TP2099

Synonym:

Target:

[Ala1,3,11,15]-Endothelin TFA

TP1512

Synonym:

Target:

Endothelin 3 (Rat,Human) (TFA)

TP1173

Synonym: Endothelin-3, human, mouse, rabbit, rat TFA

Target:

[Ala1,3,11,15]-Endothelin (53-63) (TFA)

T75772

Synonym:

Target:

Big Endothelin-1 (1-38), human

T36479

Synonym:

Target:

Endothelin-1 (1-15), amide, human

TP2246

Synonym:

Target: Others

Endothelin 1 (swine, human)

T19309

Synonym:

Target: Others

Endothelin 1 (swine, human) (TFA)

T75731

Synonym:

Target:

Endothelin-1 (1-31) (Human)

T76564

Synonym:

Target:

Endothelin 1 (swine, human), Alexa Fluor 488-labeled

T76081

Synonym:

Target:

Endothelin-1 (1-31) (Human) acetate

Ac-Endothelin-1 (16-21), human

T22540

Synonym:

Target: Others

Endothelin-3, human, mouse, rabbit, rat

TP1175

Synonym: Endothelin 3 (Rat,Human)

Target:

Big Endothelin-1 (1-39), porcine

T36480

Synonym:

Target:

Endothelin-1 (1-31) (Human) TFA

T78063

Synonym:

Target: ERK

[Asn18] Endothelin-1, human

T76329

Synonym:

Target:

Methantheline Bromide

T33314

Synonym: Frenogastrico,Dixamone bromide,Banthine,Asabaine,Methanthelinium bromide

Target:

[Ala2] Endothelin-3, human

T76305

Synonym:

Target:

Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPY-00132	Mesothelin Protein, Human, Recombinant	Human	HEK293 Cells
	Mesothelin Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 32.4 kDa and the accession number is Q13421-3.
TMPK-00961	MSLN/Mesothelin Protein, Human, Recombinant (His & Avi), FITC-Labeled	Human	HEK293 Cells
	MSLN/Mesothelin Protein, Human, Recombinant (His & Avi), FITC-Labeled is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 35.2 kDa and the accession number is Q13421-2.
TMPK-00960	MSLN/Mesothelin Protein, Human, Recombinant (His & Avi), PE-Labeled	Human	HEK293 Cells
	MSLN/Mesothelin Protein, Human, Recombinant (His & Avi), PE-Labeled is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 35.2 kDa and the accession number is Q13421-2.
TMPY-02875	Mesothelin Protein, Human, Recombinant (hFc), Biotinylated	Human	HEK293 Cells
	Mesothelin Protein, Human, Recombinant (hFc), Biotinylated is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 60.7 kDa and the accession number is Q13421-2.
TMPY-06914	Mesothelin Protein, Rat, Recombinant (His)	Rat	HEK293 Cells
	Mesothelin Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 35.48 kDa and the accession number is Q9ERA7.
TMPY-06861	Mesothelin Protein, Mouse, Recombinant (His & Avi)	Mouse	HEK293 Cells
	Mesothelin Protein, Mouse, Recombinant (His & Avi) is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 37.41 kDa and the accession number is Q61468-1.
TMPK-01377	MSLN/Mesothelin Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	MSLN/Mesothelin Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 33 kDa and the accession number is A0A2K5TW94-1.
TMPK-01368	MSLN/Mesothelin Protein, Cynomolgus, Recombinant (hFc)	Cynomolgus	HEK293 Cells
	MSLN/Mesothelin Protein, Cynomolgus, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-hFc tag. The predicted molecular weight is 58.6 kDa and the accession number is A0A2K5TW94-1.
TMPY-05129	Mesothelin Protein, Human, Recombinant (His), Biotinylated	Human	HEK293 Cells
	Mesothelin Protein, Human, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 28.2 kDa and the accession number is Q13421-2.
TMPK-01397	MSLN/Mesothelin Protein (Primary Amine Labeling), Cynomolgus, Recombinant (His), Biotinylated	Cynomolgus	HEK293 Cells
	MSLN/Mesothelin Protein (Primary Amine Labeling), Cynomolgus, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 33 kDa and the accession number is A0...
TMPY-03146	Mesothelin Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Mesothelin Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 28.2 kDa and the accession number is Q13421-2.
TMPH-01295	Endothelin-1/EDN1 Protein, Human, Recombinant (GST)	Human	E. coli
	Endothelins are endothelium-derived vasoconstrictor peptides. Probable ligand for G-protein coupled receptors EDNRA and EDNRB which activates PTK2B, BCAR1, BCAR3 and, GTPases RAP1 and RHOA cascade in glomerular mesangial...
TMPY-06904	Mesothelin Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	Mesothelin Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 33.31 kDa and the accession number is XM_005590816.3.
TMPY-06773	Mesothelin Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	Mesothelin Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 35.44 kDa and the accession number is AAH09272.1.
TMPK-00962	MSLN/Mesothelin Protein, Human, Recombinant (His & Avi)	Human	HEK293 Cells
	MSLN/Mesothelin Protein, Human, Recombinant (His & Avi) is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 35.2 kDa and the accession number is Q13421-2.
TMPY-06776	Mesothelin Protein, Human, Recombinant (hFc & Avi), Biotinylated	Human	HEK293 Cells
	Mesothelin Protein, Human, Recombinant (hFc & Avi), Biotinylated is expressed in HEK293 mammalian cells with hFc and Avi tag. The predicted molecular weight is 60.72 kDa and the accession number is AAH09272.1.
TMPY-06787	Mesothelin Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	Mesothelin Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 35.6 kDa and the accession number is Q61468-1.
TMPK-00959	MSLN/Mesothelin Protein, Human, Recombinant (hFc & Avi), Biotinylated	Human	HEK293 Cells
	MSLN/Mesothelin Protein, Human, Recombinant (hFc & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-hFc-Avi tag. The predicted molecular weight is 61.1 kDa and the accession number is Q13421-2.
TMPK-00963	MSLN/Mesothelin Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	MSLN/Mesothelin Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 35.2 kDa and the accession number is Q13421-2.
TMPY-03116	Mesothelin Protein, Human, Recombinant (aa 296-580, hFc)	Human	HEK293 Cells
	Mesothelin Protein, Human, Recombinant (aa 296-580, hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 60.7 kDa and the accession number is Q13421-2.
TMPH-03286	Endothelin-1/EDN1 Protein, Rat, Recombinant (His & KSI)	Rat	E. coli
	Endothelins are endothelium-derived vasoconstrictor peptides. Probable ligand for G-protein coupled receptors EDNRA and EDNRB which activates PTK2B, BCAR1, BCAR3 and, GTPases RAP1 and RHOA cascade in glomerular mesangial...
TMPY-03860	Endothelin B Receptor Protein, Human, Recombinant (mFc)	Human	HEK293 Cells
	Endothelin B Receptor Protein, Human, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 34.4 kDa and the accession number is P24530-1.
TMPY-02951	Mesothelin Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Mesothelin Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 53.7 kDa and the accession number is Q13421-2.
TMPK-01026	MSLN/Mesothelin Protein (Primary Amine Labeling), Mouse, Recombinant (His), Biotinylated	Mouse	HEK293 Cells
	MSLN/Mesothelin Protein (Primary Amine Labeling), Mouse, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 35.2 kDa and the accession number is Q6146...
TMPY-00181	Endothelin B Receptor Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Endothelin B Receptor Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 9.5 kDa and the accession number is P24530-1.