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T23523 |
W-5 hydrochloride
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W-5 HCl,W 5 (hydrochloride),N-(6-Aminohexyl)-1-naphthalenesulfonamide HCl |
CaMK
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W-5 hydrochloride (N-(6-Aminohexyl)-1-naphthalenesulfonamide HCl) is a potent calmodulin antagonist. |
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T23525 |
W-9 hydrochloride
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N-(6-aminohexyl)-5-chloronaphthalene-2-sulfonamide hydrochloride |
CaMK
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W-9 hydrochloride is a calmodulin antagonist. |
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T20792 |
W-7 hydrochloride
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W 7 HCl,W7 HCl,W-7 HCl |
CaMK
,
Apoptosis
,
Myosin
,
PDE
|
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W-7 hydrochloride (W-7 HCl), a calmodulin antagonist, inhibits Ca2+-calmodulin-dependent myosin light chain kinase and phosphodiesterase, W-7 hydrochloride induces apoptosis and has antitumor activity. |
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T26911 |
Bromotetrandrine
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5-Bromotetrandrine,W-198,BrTet,W 198,W198 |
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Bromotetrandrine is an P-glycoprotein inhibitor, which were developed and coadministered with chemotherapeutic drugs to overcome the effect of efflux pumps thus enhancing the chemosensitivity of therapeutics. |
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TNU1235 |
N4-Benzoyl-5'-O-DMT-5-methylcytidine
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Nucleoside Derivatives - Protected nucleosides w/NH2/OH open |
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TNU1365 |
2'-Deoxy-5'-O-DMT-5-methylcytidine
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2'-Deoxy-5'-O-DMT-5-methylcytidine is a Nucleoside Derivative - Protected nucleoside w/NH2/OH open. |
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TNU1413 |
5’-O-(4,4-Dimethoxytrityl)-3’-deoxy-5-methyluridine
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5'-O-(4,4-Dimethoxytrityl)-3'-deoxy-5-methyluridine is a Nucleoside Derivative - Protected nucleoside w/NH2/OH open; 3'-Deoxy nucleoside. |
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TNU1385 |
5’-O-(4,4’-Dimethoxytrityl)-3’-O-(2-methoxyethyl) uridine
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5'-O-(4,4'-Dimethoxytrityl)-3'-O-(2-methoxyethyl) uridine is a Nucleoside Derivative - 3'-Modified nucleoside; Protected nucleoside w/NH2/OH open. |
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TNU1445 |
5’-(4,4’-Dimethoxytrityl)-5-methyluridine
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5'-(4,4'-Dimethoxytrityl)-5-methyluridine is a Nucleoside Derivative - Protected nucleoside w/NH2/OH open. |
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TNU1284 |
3’-O-(t-Butyldimethylsilyl)-2’-O-(2-methoxyethyl)-5-methyluridine
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3'-O-(t-Butyldimethylsilyl)-2'-O-(2-methoxyethyl)-5-methyluridine is a Nucleoside Derivative - Protected nucleoside w/NH2/OH open; 2'-Modified nucleoside. |
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TNU1376 |
N2-iso-Butyroyl-5'-O-DMT-3'-deoxy-3'-fluoroguanosine
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N2-iso-Butyroyl-5'-O-DMT-3'-deoxy-3'-fluoroguanosine is a Nucleoside Derivative - Fluoro-modified nucleoside; Protected nucleoside w/NH2/OH open. |
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TNU1298 |
N4-Benzoyl-2'-deoxy-5'-O-DMT-2',2'-difluorocytidine
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|
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N4-Benzoyl-2'-deoxy-5'-O-DMT-2',2'-difluorocytidine is a Nucleoside Derivative - Fluoro-modified nucleoside; Protected nucleoside w/NH2/OH open. |
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TNU1076 |
5’-O-Acetyl-5-acetyloxymethyluridine
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|
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Nucleoside Derivatives - 5-Modified pyrimidine nucleosides; Protected nucleosides w/NH2/OH open |
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TNU1383 |
N2-iso-Butyroyl-5’-O-(4,4’-dimethoxytrityl)-3’-O-Methyl guanosine
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N2-iso-Butyroyl-5'-O-(4,4'-dimethoxytrityl)-3'-O-Methyl guanosine is a Nucleoside Derivative - 3'-Modified nucleoside; Protected nucleoside w/NH2/OH open. |
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TNU1362 |
N4-Benzoyl-5’-O-DMT-3’-O-(2-methoxyethyl)-5-methylcytidine
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N4-Benzoyl-5'-O-DMT-3'-O-(2-methoxyethyl)-5-methylcytidine is a Nucleoside Derivative - 3'-Modified nucleoside; Protected nucleoside w/NH2/OH open. |
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TNU1378 |
5’-O-(4,4’-Dimethoxytrityl)-3’-O-methyluridine
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|
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5'-O-(4,4'-Dimethoxytrityl)-3'-O-methyluridine is a Nucleoside Derivative - 3'-Modified nucleoside; Protected nucleoside w/NH2/OH open. |
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TNU0045 |
β-D-Ribofuranose analogue 1
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Nucleoside Derivatives - 5-Modified pyrimidine nucleosides; Thio-nucleosides; Amino nucleosides; Protected nucleosides w/NH2/OH open |
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TNU1390 |
N2-iso-Butyroyl-5’-O-DMT-3’-O-(methoxyethyl)guanosine
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|
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N2-iso-Butyroyl-5'-O-DMT-3'-O-(methoxyethyl)guanosine is a Nucleoside Derivative - 3'-Modified nucleoside; Protected nucleoside w/NH2/OH open. |
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TNU1416 |
N4-Benzoyl-5’-O-(4,4-dimethoxytrityl)-3’-deoxycytidine
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N4-Benzoyl-5'-O-(4,4-dimethoxytrityl)-3'-deoxycytidine is a Nucleoside Derivative - Protected nucleoside w/NH2/OH open; 3'-Deoxy nucleoside. |
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TNU1323 |
3’,5’-Bis(O-t-butyldimethylsilyl)-4’-C-hydroxymethyl thymidine
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3',5'-Bis(O-t-butyldimethylsilyl)-4'-C-hydroxymethyl thymidine is a Nucleoside Derivative - 4'-Modified nucleoside; Protected nucleoside w/NH2/OH open. |
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T76186 |
Tyr-W-MIF-1
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Tyr-W-MIF-1, an opioid tetrapeptide, exhibits both opiate and antiopiate activities, and has been demonstrated to induce analgesia [1] [2] [5]. |
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T14359 |
AVX 13616
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Others
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AVX 13616, Avexa's leading antibacterial candidate, demonstrates significant in vivo antibacterial efficacy, especially against drug-resistant Staphylococcus pathogens, with an IC50 value of 2-4 µg/ml (MICs) and is targe... |
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T1087L |
Valaciclovir
|
|
|
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Valacyclovir (Valaciclovir) is an orally active antiviral drug for herpes simplex, herpes zoster, and herpes B. Valacyclovir inhibits HSV-1 W with an IC50 of 2.9 μg/ml. Valacyclovir is a prodrug of Aciclovir [1] [2] [3] ... |
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T36379 |
Halometasone
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|
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Halometasone is a synthetic corticosteroid.1,2Formulations containing halometasone have been used in the treatment of psoriasis vulgaris and eczematous dermatoses.
1.de la Brassine, M., Kint, A., Lachapelle, J.M., et al.... |
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T36986 |
Colletodiol
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Colletodiol is a fungal metabolite that has been found inD. grovesiiand has immunosuppressant and antiviral activities.1,2It inhibits concanavalin A- or LPS-induced proliferation of isolated mouse splenocytes (IC50s = 12... |
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T36916 |
Estrone-3-Glucuronide (sodium salt hydrate)
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Estrone-3-Glucuronide is a metabolite of the primary premenopausal estrogen 17β-estradiol .1,2Urinary levels of estrone-3-Glucuronide peak approximately 36 hours prior to ovulation and have been used as a marker of ferti... |
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T35513 |
13C15-Nivalenol
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13C15-Nivalenol |
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13C15-Nivalenol is intended for use as an internal standard for the quantification of nivalenol by GC- or LC-MS. Nivalenol is a trichothecene mycotoxin that has been found inFusarium.1It is lethal to mice (LD50= 6.9 mg/k... |
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T36974 |
D-threo-PPMP hydrochloride
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D-threo-PPMP is a glucosylceramide (GlyCer) synthetase inhibitor.1,2It is the active enanantiomer and enzymatic inhibitory component of the racemic DL-threo-PPMP . In MDCK kidney epithelial cells, D-threo-PPMP induces a ... |
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T37248 |
Pantothenate Kinase Inhibitor
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|
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Pantothenate Kinase Inhibitor (PANKi) is a reversible inhibitor of pantothenate kinase (PanK; IC50s = 70, 92, and 25 nM for PanK1β, PanK2, and PanK3, respectively), the rate-limiting enzyme in the synthesis of coenzyme A... |
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T37347 |
6'-Sialyllactose Sodium Salt
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6'-Sialyllactose Sodium Salt,6'-N-Acetylneuraminyl-D-lactose |
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6'-Sialyllactose consists of the monosaccharide N-acetylneuraminic acid linked to the galactosyl subunit of lactose at the 6 position. This connection is at the 3 position in the related compound, 3’-sialyllactose. Both ... |
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T35683 |
2-deoxy-D-Glucose-13C6
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2-deoxy-D-Glucose-13C6 |
|
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2-deoxy-D-Glucose-13C6is intended for use as an internal standard for the quantification of 2-deoxy-D-glucose by GC- or LC-MS. 2-deoxy-D-Glucose is a glucose antimetabolite and an inhibitor of glycolysis.1,2It inhibits h... |
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T35955 |
PAR2 (1-6) amide (human) (trifluoroacetate salt)
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PAR2 (1-6) amide (human) (trifluoroacetate salt) |
|
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PAR2 (1-6) amide is a synthetic peptide agonist of proteinase-activated receptor 2 (PAR2) that corresponds to residues 1-6 of the amino terminal tethered ligand sequence of human PAR2 and residues 37-42 of the full-lengt... |
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T36521 |
Alaproclate (hydrochloride)
|
|
|
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Alaproclate is a selective serotonin reuptake inhibitor (SSRI).1,2 It inhibits depletion of serotonin (5-HT) induced by 4-methyl-α-ethyl-m-tyramine in rat cerebral cortex, hippocampus, hypothalamus, and striatum (EC50s =... |
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T35451 |
β-Defensin-2 (human) (trifluoroacetate salt)
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β-Defensin-2 is a peptide with antimicrobial properties that protects the skin and mucosal membranes of the respiratory, genitourinary, and gastrointestinal tracts.1It inhibits the growth of periodontopathogenic and cari... |
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T35426 |
β-Defensin-1 (human) (trifluoroacetate salt)
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β-Defensin-1 is a peptide with antimicrobial properties that protects the skin and mucosal membranes of the respiratory, genitourinary, and gastrointestinal tracts.1It inhibits the growth ofB. adolescentis,L. acidophilus... |
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T35775 |
HT-2 Toxin-13C22
|
HT-2 Toxin-13C22 |
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HT-2 toxin-13C22is intended for use as an internal standard for the quantification of HT-2 toxin by GC- or LC-MS. HT-2 toxin is a type A trichothecene mycotoxin and an active, deacetylated metabolite of the trichothecene... |
