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T9626 |
Cycloleucine
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NMDAR
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Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM. Cycloleucine is also a competitive inhibitor of S-adenosyl-methionine mediated methylation with anxiolytic and cytostatic ef... |
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T27112 |
Cytembena
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DNA/RNA Synthesis
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Cytembena is a cytostatic and a carcinogenic compound that may increase the incidence of fibroadenomas.Cytembena broadly inhibits DNA biosynthesis. |
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T13569 |
Benin
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Butocine,Butocin |
Others
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Benin (Butocine) is an effective cytostatic drug used for the treatment of generalized carcinoma of the breast. |
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T14871 |
Carboxyamidotriazole Orotate
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L-651582 Orotate,CAI Orotate |
Calcium Channel
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Carboxyamidotriazole Orotate (L-651582 Orotate) is a cytostatic inhibitor of non-voltage-operated calcium channels and calcium channel-mediated signaling pathways. Carboxyamidotriazole Orotate (L-651582 Orotate) is the o... |
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T35057 |
Vinformide
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NS269419,Formyl-leurosine,NSC 269419,NSC-269419 |
Others
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Vinformide is a potent cytostatic agent. |
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T40603 |
Dihydrochlamydocin
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Others
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Dihydrochlamydocin, an inhibitor of histone deacetylases (HDAC), exhibits potent cytostatic activity against mastocytoma cells. |
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T68666 |
Benfluron Hydrochloride
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Others
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Benfluron Hydrochloride is an inhibitor of HIV-1 Rev function which also acts as a cytostatic agent with substantial antiretroviral activity. |
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T14872 |
Carboxyamidotriazole
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CAI,L-651582 |
Calcium Channel
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Carboxyamidotriazole is a cytostatic inhibitor of non-voltage-operated calcium channels and calcium channel-mediated signaling pathways. It shows anti-inflammatory, anti-tumor, and antiangiogenic effects. |
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T71063 |
Tolytoxin
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Others
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Tolytoxin is a cytostatic, antifungal macrolide produced by blue-green algae of the genus Scytonema, is a potent, reversible inhibitor of cytokinesis in cultured mammalian cells |
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T23697 |
AL-8417
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J1.090.276B,AL8417,(2R)-AL-5898 |
Others
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AL-8417 is an enzyme inhibitor. It acting as an antioxidant, anti-inflammatory, and cytostatic agent. It also has the ability to suppress vitrectomy-induced posterior lens fiber changes. |
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T24258 |
KCG 1
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KCG-1,KCG1 |
Others
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KCG 1 is a keto-C-glycoside drug with antiproliferative and cytotoxic properties on tumor cells. KCG1 was 25-125 times more cytostatic on epithelial cells than on lymphoma. |
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T25043 |
Alestramustine
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Others
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Alestramustine is a cytostatic antineoplastic agent. The drug, via its active metabolites, binds to microtubule-associated proteins and β-tubulin and interferes with microtubule function, thereby suppressing cell divisio... |
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T13889 |
SLLN-15
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Others
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SLLN-15 is an oral active, selective and potent enhancer of autophagy. SLLN-15 activates cytostatic macroautophagy/autophagy in triple-negative breast cancer (TNBC) [1]. |
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T60401 |
Tezacitabine
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Others
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Tezacitabine is a cytostatic and cytotoxic antimetabolite. Tezacitabine is a nucleoside analogue characterized by a dual mechanism of action. Tezacitabine irreversibly inhibits ribonucleotide reductase and can be incorpo... |
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T69117 |
Pinafide
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Others
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Pinafide is a rodenticide and anti-protozoal agent. Pinafide shows strong cytostatic activity against both HeLa and KB cells and is moderately toxic to both mice and rats. It has been proved active against experimental t... |
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T75142 |
Acid Ceramidase-IN-2
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Others
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Acid Ceramidase-IN-2 (compound 1), an acid ceramidase inhibitor, exhibits potentially antiproliferative and cytostatic effects. This compound is of interest due to the overexpression of human acid ceramidase in prostate ... |
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T36107 |
YW3-56
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YW3-56 |
Others
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YW3-56 is a potent peptidylarginine deiminase (PAD) inhibitor, with an IC50 of 1-5 μM for PAD4.
Compared with Cl-amidine, YW3-56 shows >60-fold increase in cell growth inhibition efficacy (IC50 about 2.5 μM) but only 5-f... |
