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Search Results for " theophylline "

ターゲット

阻害剤

天然化合物

カタログ番号	製品名	別名	ターゲット
T1083L	Theophylline monohydrate	Quibron	HDAC , PDE , Adenosine Receptor
	Theophylline monohydrate (Quibron) appears to inhibit phosphodiesterase and prostaglandin production, regulate calcium flux and intracellular calcium distribution, and antagonize adenosine. Theophylline monohydrate is a ...		HDAC , PDE , Adenosine Receptor
T33062	Lysine theophylline
	Lysine theophylline is a soluble theophylline.
T71329	Theophylline-d6
	Theophylline-d6 is intended for use as an internal standard for the quantification of theophylline by GC- or LC-MS. Theophylline is an inhibitor of phosphodiesterase. It is also an adenosine A1 and A2 receptor antagonist...
T0829	Etofylline	7-(β-Hydroxyethyl)theophylline,Aethophyllinum,7-Theophyllineethanol,Oxyphylline,Cordalin	Others
	Etofylline (Oxyphylline) is used for difficulty in breathing, asthma, breathing difficulty and other conditions.		Others
T34839	Theophylline, 7-ethyl-6-thio-
	Theophylline, 7-ethyl-6-thio- is a bioactive chemical.
T60511	Theophylline sodium glycinate
	Theophylline (1,3-Dimethylxanthine) sodium glycinate is a potent inhibitor of phosphodiesterase (PDE) that inhibits PDE3 activity to relax airway smooth muscle. Theophylline sodium glycinate can be used for the research ...
T34837	Theophylline, 7-(2-(diethylamino)ethyl)-6-thio-, methiodide
	Theophylline, 7-(2-(diethylamino)ethyl)-6-thio-, methiodide is a bioactive chemical.
T34836	Theophylline, 7-(2-(diethylamino)ethyl)-6-thio-, hydrochloride
	Theophylline, 7-(2-(diethylamino)ethyl)-6-thio-, hydrochloride is a bioactive chemical.
T34838	Theophylline, 7-(2-oxo-4-piperidinobutyl)-6-thio-, hydrochloride
	Theophylline, 7-(2-oxo-4-piperidinobutyl)-6-thio-, hydrochloride is a bioactive chemical.
T32803	LJ 278	LJ-278,p-Dimethylamino-benzyl theophylline chlorhydrate,LJ278
	LJ-278 is a bioactive chemical.
T8634	8-Bromotheophylline	Bromotheophylline	Others
	8-Bromotheophylline (Bromotheophylline) is the active moiety of pamabrom, a mixture of 2-amino-2-methyl-propanol and bromotheophylline. From this mixture, 8-Bromotheophylline acts as a weak diuretic that has been used al...		Others
TMIH-0064	8-Chlorotheophylline-d6
	8-Chlorotheophylline-d6 is a deuterated compound of 8-Chlorotheophylline. 8-Chlorotheophylline has a CAS number of 85-18-7.
T14958	Choline theophyllinate	Oxtriphylline	Endogenous Metabolite , PDE
	Choline theophyllinate (Oxtriphylline) is the choline salt of theophylline, a small molecule PDE inhibitor that can be used to treat immune system disorders and respiratory disorders, and to study asthma disorders.		Endogenous Metabolite , PDE
T9319	Tosufloxacin	tosufloxacin tosilate,Ozex,7-(3-Aminopyrrolidin-1-yl)-1-(2,4-difluorophenyl)-6-fluoro-4-oxo-1,8-naphthyridine-3-carboxylic acid	Others
	Tosufloxacin (Ozex) is a quinolone antimicrobial agent and potent inhibitor of the metabolism of theophylline.		Others
T30686L	Cafedrine HCl	Cafedrine hydrochloride,Akrinor,L-Net
	Cafedrine HCl is a chemical linkage of norephedrine and theophylline.
T31432	Dicarboxidine
	Dicarboxidine can be used in immunochromatographic assay of theophylline in whole blood.
T40907	Theophyllol
	Theophyllol (theophylline sodium acetate) can alter calcium levels in subcellular fractions of rat brain cortex.
T39485	NCT-501 hydrochloride
	NCT-501 hydrochloride is a highly potent and selective inhibitor of aldehyde dehydrogenase 1A1 (ALDH1A1), which is based on theophylline. It effectively inhibits hALDH1A1 with an IC50 value of 40 nM, exhibiting superior ...
T70974	Cipamfylline
	Cipamfylline is a xanthine, a theophylline analogue, and is a potent and selective inhibitor of phosphodiesterase type 4 (PDE-4). Cipamfylline was tested in patients with a diagnosis of atopic dermatitis and in two human...
T70097	Acefylline piperazine
	Acefylline piperazine is a stimulant drug of the xanthine chemical class. It acts as an adenosine receptor antagonist. Acephylline piperazine is a theophylline derivative with a direct bronchodilator action. It has the a...
T60461	Ambuphylline
	Ambuphylline (Bufylline) is a theophylline derivative that may act by inhibiting phosphodiesterase. Ambuphylline is a bronchodilator that can be used in asthma and other lung disease research [1].

Compounds

Theophylline monohydrate

T1083L

Synonym: Quibron

Target: HDAC, PDE, Adenosine Receptor

Lysine theophylline

Synonym: 7-(β-Hydroxyethyl)theophylline,Aethophyllinum,7-Theophyllineethanol,Oxyphylline,Cordalin

Target: Others

Theophylline, 7-ethyl-6-thio-

T34839

Synonym:

Target:

Theophylline sodium glycinate

T60511

Synonym:

Target:

Theophylline, 7-(2-(diethylamino)ethyl)-6-thio-, methiodide

T34837

Synonym:

Target:

Theophylline, 7-(2-(diethylamino)ethyl)-6-thio-, hydrochloride

T34836

Synonym:

Target:

Theophylline, 7-(2-oxo-4-piperidinobutyl)-6-thio-, hydrochloride

Synonym: LJ-278,p-Dimethylamino-benzyl theophylline chlorhydrate,LJ278

Target:

8-Bromotheophylline

T8634

Synonym: Bromotheophylline

Target: Others

8-Chlorotheophylline-d6

TMIH-0064

Synonym:

Target:

Choline theophyllinate

T14958

Synonym: Oxtriphylline

Target: Endogenous Metabolite, PDE

Tosufloxacin

T9319

Synonym: tosufloxacin tosilate,Ozex,7-(3-Aminopyrrolidin-1-yl)-1-(2,4-difluorophenyl)-6-fluoro-4-oxo-1,8-naphthyridine-3-carboxylic acid

Target: Others

Cafedrine HCl

T30686L

Synonym: Cafedrine hydrochloride,Akrinor,L-Net

NCT-501 hydrochloride

Acefylline piperazine

カタログ番号	製品名	別名	ターゲット
T1083	Theophylline	Theo-24,1,3-Dimethylxanthine	Endogenous Metabolite , HDAC , PDE , Adenosine Receptor , Autophagy
	Theophylline (1,3-Dimethylxanthine) is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and central nervous system stimulant activities. Theophylline inhibits the 3...
T5940	Proxyphylline	7-(2-Hydroxypropyl)theophylline	PDE , Adenosine Receptor
	Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor. Proxyphylline acts as a cardiac stimulant, vasodilator and bronchodilator.		PDE , Adenosine Receptor
T2205	Acefylline	Theophylline-7-acetic acid,Carboxymethyltheophylline,acetyloxytheophylline,Theophyllineacetic acid	TNF , PAD , PKA , HDAC , PDE , Adenosine Receptor
	Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist. It is combined with diphenhydramine in the pharmaceutical preparation Etanautine to help...		TNF , PAD , PKA , HDAC , PDE , Adenosine Receptor
T10021	1-Methylxanthine		Endogenous Metabolite
	1-Methylxanthine is a caffeine derivative. 1-Methylxanthine is an essential human urinary metabolite of caffeine and theophylline (1,3-dimethylxanthine, TP). 1-Methylxanthine enhances the radiosensitivity of tumor cells.		Endogenous Metabolite
T8075	1,3-Dimethyluric acid		Endogenous Metabolite
	1,3-Dimethyluric acid is a product of theophylline metabolism in man. It is one of the purine components in urinary calculi.		Endogenous Metabolite
T0480	Doxofylline	Doxophylline	PDE , Adenosine Receptor
	Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7. As a drug used in the treatment of asthma, doxofylline has shown similar efficacy to theophylline but with s...		PDE , Adenosine Receptor
TN6339	(R)-5-Hydroxy-1,7-diphenylheptan-3-one	(5R)-Dihydroyashabushiketol	Others
	(R)-5-Hydroxy-1,7-diphenylheptan-3-one ((5R)-Dihydroyashabushiketol) is extracted from the rhizomes of Alpinia officinarum, a Chinese medicinal herb. (R)-5-Hydroxy-1,7-diphenylheptan-3-one inhibits melanogenesis in theop...		Others
TN1486	Chimonanthine		Others
	(-)-Chimonanthine (IC50 = 0.93 μM) shows potent inhibitory effects on melanogenesis in theophylline-stimulated murine B16 melanoma 4A5 cells.		Others