Adenosine Receptor

The adenosine receptors are a class of purinergic G protein-coupled receptors with adenosine as the endogenous ligand. There are four known types of adenosine receptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene.

Cat. No.	製品名	CAS No.	Purity
T15418	GS-6201	752222-83-6	98%
T15418	GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors with a ...
T21620	Adenosine receptor antagonist 4	133240-06-9	98%
T21620	Adenosine receptor antagonist 4 is an adenosine receptor antagonist.
T16140	MRS 1754	264622-58-4	98%
T16140	MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.
T12107	MRS-3777 hemioxalate	1186195-57-2	98%
T12107	MRS-3777 hemioxalate is a selective adenosine A3 receptor antagonist that reverses the anti-injury perception effects of its corresponding agonist and can be use...
T14078	AB928	2239273-34-6	98%
T14078	AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].
T7188	Piclidenoson	152918-18-8	98%
T7188	Piclidenoson (CF-101), a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust anti-inflammatory effect in psoriasis patients.
T16782	Rolofylline	136199-02-5	98%
T16782	Rolofylline (KW-3902) is a selective adenosine A1 receptor antagonist used in the study of acute congestive heart failure and renal dysfunction, and in the study...
T7320	Tozadenant	870070-55-6
T7320	Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)
T0070	Pentoxifylline	6493-05-6
T0070	Pentoxifylline (PTX) modulates immunologic activity by stimulating cytokine production. Pentoxifylline is a methylxanthine derivative that inhibits phosphodieste...
T4668	ABT-702 dihydrochloride	1188890-28-9
T4668	ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.
T0480	Doxofylline	69975-86-6
T0480	Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7. As a drug used in the treatment of asthma, doxofy...
T8613	1-Ethyl-6-aminouracil	41862-09-3
T8613	1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high affi...
T29112	VPC171	1018830-99-3
T29112	VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).
T72067	DPTN dihydrochloride	325767-87-1	100%
T72067	DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.
T15715	LAS101057	925676-48-8	100%
T15715	LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.
T9180	LUF6096	1116652-18-6	100%
T9180	LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically while demonstr...
T0665	Xanthine	69-89-6	89.06%
T0665	Xanthine (Isoxanthine) is a product on the pathway of purine degradation. Xanthine is subsequently converted to uric acid by the action of the Xanthine oxidase e...
T27076	8-Cyclopentyl-1,3-dimethylxanthine	35873-49-5	95.00%
T27076	8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.
T14127	Adenosine A1 receptor activator T62	40312-34-3	95.00%
T14127	Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also r...
T7021	ZM241385	139180-30-6	95.28%
T7021	ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.