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Adenosine Receptor

The adenosine receptors are a class of purinergic G protein-coupled receptors with adenosine as the endogenous ligand. There are four known types of adenosine receptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene.
Cat. No. 製品名 CAS No. Purity Chemical Structure
T7320 Tozadenant 870070-55-6 98%
Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)
T0070 Pentoxifylline 6493-05-6 98%
Pentoxifylline (PTX) modulates immunologic activity by stimulating cytokine production. Pentoxifylline is a methylxanthine derivative that inhibits phosphodieste...
T4668 ABT-702 dihydrochloride 1188890-28-9 98%
ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.
T21017 5'-Amino-5'-deoxyadenosine 14365-44-7 98%
5'-Amino-5'-deoxyadenosine (NH2dAdo) is an adenosine kinase inhibitor targeting malignant tumors of the inert lymphatic system with antitumor and anticancer effe...
T4290 Preladenant 377727-87-2 98%
Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosine ...
T15418 GS-6201 752222-83-6 98%
GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors with a ...
T0480 Doxofylline 69975-86-6 98%
Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7. As a drug used in the treatment of asthma, doxofy...
T16378 Ogerin 1309198-71-7 98%
Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83). Ogerin blocks recall in fear conditioning in mice. Ogerin displays inverse agonist and a...
T21620 Adenosine receptor antagonist 4 133240-06-9 98%
Adenosine receptor antagonist 4 is an adenosine receptor antagonist.
T14078 AB928 2239273-34-6 98%
AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].
T7188 Piclidenoson 152918-18-8 98%
Piclidenoson (CF-101), a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust anti-inflammatory effect in psoriasis patients.
T27076 8-Cyclopentyl-1,3-dimethylxanthine 35873-49-5 98%
8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.
T22489 2'-MeCCPA 205171-12-6 98%
2'-MeCCPA is a potent and highly selective A1 adenosine receptor (A1AR) agonist with a K-value of 1.8 nM for AR.2'-MeCCPA inhibits trichostatin-stimulated adenyl...
T34914 Trabodenoson 871108-05-3 98%
Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.
T15715 LAS101057 925676-48-8 98%
LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.
T29112 VPC171 1018830-99-3 98%
VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).
T16263 N6-Cyclopentyladenosine 41552-82-3 98%
N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's of ...
T8613 1-Ethyl-6-aminouracil 41862-09-3
1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high affi...
T72067 DPTN dihydrochloride 325767-87-1 100%
DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.
T10248 Adenosine antagonist-1 431040-19-6 100%
Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.
Tozadenant
T7320
Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)
Pentoxifylline
T0070
Pentoxifylline (PTX) modulates immunologic activity by stimulating cytokine production. Pentoxifylline is a methylxanthine derivative that inhibits phosphodieste...
ABT-702 dihydrochloride
T4668
ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.
5'-Amino-5'-deoxyadenosine
T21017
5'-Amino-5'-deoxyadenosine (NH2dAdo) is an adenosine kinase inhibitor targeting malignant tumors of the inert lymphatic system with antitumor and anticancer effe...
Preladenant
T4290
Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosine ...
GS-6201
T15418
GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors with a ...
Doxofylline
T0480
Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7. As a drug used in the treatment of asthma, doxofy...
Ogerin
T16378
Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83). Ogerin blocks recall in fear conditioning in mice. Ogerin displays inverse agonist and a...
Adenosine receptor antagonist 4
T21620
Adenosine receptor antagonist 4 is an adenosine receptor antagonist.
AB928
T14078
AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].
Piclidenoson
T7188
Piclidenoson (CF-101), a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust anti-inflammatory effect in psoriasis patients.
8-Cyclopentyl-1,3-dimethylxanthine
T27076
8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.
2'-MeCCPA
T22489
2'-MeCCPA is a potent and highly selective A1 adenosine receptor (A1AR) agonist with a K-value of 1.8 nM for AR.2'-MeCCPA inhibits trichostatin-stimulated adenyl...
Trabodenoson
T34914
Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.
LAS101057
T15715
LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.
VPC171
T29112
VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).
N6-Cyclopentyladenosine
T16263
N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's of ...
1-Ethyl-6-aminouracil
T8613
1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high affi...
DPTN dihydrochloride
T72067
DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.
Adenosine antagonist-1
T10248
Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.
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