Powder: -20°C for 3 years | In solvent: -80°C for 1 year
GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors with a Ki of 22 nM.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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1 mg | 在庫あり | ¥ 8,500 | |||
5 mg | 在庫あり | ¥ 22,000 | |||
10 mg | 在庫あり | ¥ 35,500 | |||
25 mg | 在庫あり | ¥ 75,500 | |||
50 mg | 在庫あり | ¥ 120,000 | |||
100 mg | 在庫あり | ¥ 174,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 27,000 |
説明 | GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors with a Ki of 22 nM. |
ターゲット&IC50 | A2B:22 nM(Ki, human), A3:1070 nM(Ki, human), A1:1940 nM(Ki, human), A2A:3280 nM(Ki, human) |
別名 | CVT-6883 |
分子量 | 446.43 |
分子式 | C21H21F3N6O2 |
CAS No. | 752222-83-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 30 mg/ml (67.2 mM), Sonication and heating to 60℃ are recommended.
You can also refer to dose conversion for different animals. 詳細
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GS-6201 752222-83-6 GPCR/G Protein Neuroscience Adenosine Receptor GS 6201 GS6201 Inhibitor remodeling cardiac caspase-1 reactivity airway affinity infarction P1 receptor CVT-6883 inhibit CVT6883 acute CVT 6883 selectivity myocardial inhibitor