Powder: -20°C for 3 years | In solvent: -80°C for 1 year
BD 1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM). BD 1008 dihydrobromide have high affinity for sigma1 receptors, moderate affinity for sigma2 receptors.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 42,000 | |||
5 mg | 在庫あり | ¥ 72,500 | |||
10 mg | 在庫あり | ¥ 113,500 | |||
25 mg | 在庫あり | ¥ 165,000 | |||
50 mg | 在庫あり | ¥ 217,000 | |||
100 mg | 在庫あり | ¥ 323,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 83,500 |
説明 | BD 1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM). BD 1008 dihydrobromide have high affinity for sigma1 receptors, moderate affinity for sigma2 receptors. |
ターゲット&IC50 | σ1:2 nM(Ki) |
分子量 | 463.08 |
分子式 | C15H24Br2Cl2N2 |
CAS No. | 138356-09-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 32.5 mg/mL (70.18 mM)
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
BD 1008 dihydrobromide 138356-09-9 GPCR/G Protein Sigma receptor BD1008 Dihydrobromide BD-1008 BD-1008 Dihydrobromide BD1008 BD 1008 BD 1008 Dihydrobromide Inhibitor inhibitor inhibit