Powder: -20°C for 3 years | In solvent: -80°C for 1 year
BP 897 (2-Naphthalenecarboxamide, N-[4-[4-(2-methoxyphenyl)-1-piperazinyl]butyl]-) is a potent and selective dopamine D3 receptor agonist, and a weak dopamine D2 receptor antagonist, with Kis of 0.92 nM and 61 nM for D3 and D2 receptors, and shows low affinities at D1 and D4 receptors (Kis, 3 and 0.3 μM, respectively).
説明 | BP 897 (2-Naphthalenecarboxamide, N-[4-[4-(2-methoxyphenyl)-1-piperazinyl]butyl]-) is a potent and selective dopamine D3 receptor agonist, and a weak dopamine D2 receptor antagonist, with Kis of 0.92 nM and 61 nM for D3 and D2 receptors, and shows low affinities at D1 and D4 receptors (Kis, 3 and 0.3 μM, respectively). |
ターゲット&IC50 | D1:3 µM (Ki), D4:0.3 µM (Ki), D3:0.92 nM (Ki), D2:61 nM (Ki) |
別名 | 2-Naphthalenecarboxamide, N-[4-[4-(2-methoxyphenyl)-1-piperazinyl]butyl]- |
分子量 | 417.54 |
分子式 | C26H31N3O2 |
CAS No. | 192384-87-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 55 mg/mL (131.72 mM)
You can also refer to dose conversion for different animals. 詳細
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BP 897 192384-87-5 GPCR/G Protein Neuroscience Dopamine Receptor inhibit cocaine drug-seeking BP-897 Inhibitor addiction behaviour motivational stimuli BP897 rewarding 2-Naphthalenecarboxamide, N-[4-[4-(2-methoxyphenyl)-1-piperazinyl]butyl]- inhibitor