Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Benzbromarone (Desuric) is a CYP2C9 inhibitor with Ki value of 19.3 nM.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
50 mg | 在庫あり | ¥ 7,500 | |||
100 mg | 在庫あり | ¥ 11,000 | |||
200 mg | 在庫あり | ¥ 14,000 | |||
500 mg | 在庫あり | ¥ 22,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 11,000 |
説明 | Benzbromarone (Desuric) is a CYP2C9 inhibitor with Ki value of 19.3 nM. |
ターゲット&IC50 | CYP2C9:19.3 nM(Ki) |
In vivo | In oocytes expressing URAT1 (IC50 <0.1 μM), Benzbromarone (50 μM) completely inhibited the uptake of uric acid. In rat hepatocytes, Benzbromarone (100 μM) increased mitochondrial size and induced apoptosis in 11% of cells. |
別名 | Desuric, Normurat, Urinorm |
分子量 | 424.08 |
分子式 | C17H12Br2O3 |
CAS No. | 3562-84-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ethanol: 9 mg/mL (21.22 mM)
DMSO: 79 mg/mL (186.3 mM)
H2O: < 1 mg/mL (insoluble or slightly soluble)
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Benzbromarone 3562-84-3 Apoptosis Metabolism Xanthine Oxidase P450 inhibit Desuric Normurat Inhibitor Urinorm inhibitor