Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).
説明 | CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM). |
ターゲット&IC50 | GABAB:85 nM |
キナーゼ試験 | Reactions are set up with Acetyl coenzyme A (AcCoA)(0.4 μM), N-terminal histone H4 peptide (sequence SGRGKGGKGLGKGGAKRHRKV-GGK-biotin)(50 nM), MOZ enzyme(10 nM), and an acetyl-lysine specific antibody (final dilution 1: 10000). |
別名 | CGP 52432 |
分子量 | 384.24 |
分子式 | C15H24Cl2NO4P |
CAS No. | 139667-74-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 5 mg/mL (13.01 mM), Sonication and heating are recommended.
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
CGP52432 139667-74-6 Membrane transporter/Ion channel Neuroscience GABA Receptor Inhibitor inhibit Gamma-aminobutyric acid Receptor CGP 52432 γ-Aminobutyric acid Receptor CGP-52432 inhibitor