store at low temperature,keep away from direct sunlight
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Camizestrant (Estrogen receptor antagonist 2) is an antagonist of the estrogen receptor and can be used in studies about ER+ HER2-advanced breast cancer[1].
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 36,500 |
5 mg | 在庫あり | ¥ 91,000 |
10 mg | 在庫あり | ¥ 152,000 |
25 mg | 在庫あり | ¥ 268,500 |
50 mg | 約6-8 週間 | ¥ 431,500 |
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 95,500 |
説明 | Camizestrant (Estrogen receptor antagonist 2) is an antagonist of the estrogen receptor and can be used in studies about ER+ HER2-advanced breast cancer[1]. |
ターゲット&IC50 | ERR: |
In vivo | In human parental MCF7 mice xenograft, oral administration of Camizestrant (0.2-50 mg/kg) displays dose-dependent anti-tumor effects. Oral administration of Camizestrant (0.8-40 mg/kg) dose-dependently decreases the growth of the tumor[1]. |
別名 | Estrogen receptor antagonist 2 |
分子量 | 476.51 |
分子式 | C24H28F4N6 |
CAS No. | 2222844-89-3 |
store at low temperature,keep away from direct sunlight
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (104.93 mM)
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Camizestrant 2222844-89-3 Endocrinology/Hormones Estrogen Receptor/ERR Estrogen receptor antagonist 2 Inhibitor inhibitor inhibit