Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DPN (Diarylpropionitrile) is an selective agonist of estrogen receptor β (ERβ) .
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
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5 mg | 在庫あり | ¥ 7,500 | |||
10 mg | 在庫あり | ¥ 12,000 | |||
25 mg | 在庫あり | ¥ 25,000 | |||
50 mg | 在庫あり | ¥ 45,500 | |||
100 mg | 在庫あり | ¥ 81,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 13,500 |
説明 | DPN (Diarylpropionitrile) is an selective agonist of estrogen receptor β (ERβ) . |
ターゲット&IC50 | ERβ:0.85 nM (EC50) |
In vitro | DPN exhibits a 70-fold higher relative binding affinity for ERβ (18%) versus ERα (0.25%), about 80-fold higher transcriptional potency (EC50 = 0.85 nM versus 66 nM), and 170-fold higher relative potency (4.6% versus 0.025%) in transcription assays[1] |
別名 | Diarylpropionitrile |
分子量 | 239.27 |
分子式 | C15H13NO2 |
CAS No. | 1428-67-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 25 mg/mL (104.48 mM)
You can also refer to dose conversion for different animals. 詳細
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DPN 1428-67-7 Apoptosis Autophagy Endocrinology/Hormones Estrogen/progestogen Receptor Estrogen Receptor/ERR inhibit neuroprotection estrogen beta anti-inflammation receptor peptide amyloid Inhibitor anxiety-like Alzheimer's antioxidant disease behaviors Diarylpropionitrile inhibitor