Powder: -20°C for 3 years | In solvent: -80°C for 1 year
dBET57 is heterobifunctional degrader of BRD4 based on the PROTAC technology, exhibits significant degradation of BRD4BD1 with a DC50/5h of 500 nM ,and inactive on BRD4BD2
説明 | dBET57 is heterobifunctional degrader of BRD4 based on the PROTAC technology, exhibits significant degradation of BRD4BD1 with a DC50/5h of 500 nM ,and inactive on BRD4BD2 |
ターゲット&IC50 | BRD4 BD1:500 nM (DC50) |
分子量 | 699.18 |
分子式 | C34H31ClN8O5S |
CAS No. | 1883863-52-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 250 mg/mL (357.56 mM)
You can also refer to dose conversion for different animals. 詳細
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Dbet57 1883863-52-2 Chromatin/Epigenetic Epigenetic Reader Domain inhibit Dbet-57 dBET 57 Inhibitor PROTACs inhibitor