Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Didesmethyl cariprazine, a metabolite of Cariprazine, is the major cyclic active part. Didesmethyl cariprazine has a long half-life of 1-3 weeks. Cariprazine is a potent D3 preference D3/D2 receptor partial agonist of dopamine for the treatment of schizophrenia, bipolar mania, and depression, with a high affinity for d3 and d2 receptors and a moderate affinity for 5-HT 1A receptors.
説明 | Didesmethyl cariprazine, a metabolite of Cariprazine, is the major cyclic active part. Didesmethyl cariprazine has a long half-life of 1-3 weeks. Cariprazine is a potent D3 preference D3/D2 receptor partial agonist of dopamine for the treatment of schizophrenia, bipolar mania, and depression, with a high affinity for d3 and d2 receptors and a moderate affinity for 5-HT 1A receptors. |
分子量 | 399.36 |
分子式 | C19H28Cl2N4O |
CAS No. | 839712-25-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 10.2 mg/mL (25.6 mM), Sonication and heating to 80℃ are recommended.
You can also refer to dose conversion for different animals. 詳細
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Didesmethyl cariprazine 839712-25-3 GPCR/G Protein Neuroscience Dopamine Receptor 5-HT Receptor Inhibitor inhibitor inhibit