Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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サンプルについてお問い合わせ | |||||
50 mg | 在庫あり | ¥ 7,500 | |||
100 mg | 在庫あり | ¥ 10,000 | |||
500 mg | 在庫あり | ¥ 22,500 | |||
1 g | 在庫あり | ¥ 34,000 |
説明 | Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM. |
ターゲット&IC50 | D1 receptor:166 nM |
In vitro | Cidofovir inhibits human cytomegalovirus (HCMV) infection in cultured cells. Cidofovir is inhibitory to CMV plaque formation even when added to the cells at 48 hr post infection with IC50 of 0.9 μg/mL for Davis and 1.6 μg/mL for AD-169 strains,respectively. [1] Cidofovir also inhibits herpes simplex virus infection. In addition, Cidofovir blocks cell fusion induced by HSV-1 in monkey kidney cells and blocks the expression of HSV-l-specific proteins and the synthesis of viral DNA. [3] |
植物由来 |
別名 | Gindarine, L-Tetrahydropalmatine, Caseanine, (-)-Tetrahydropalmatine |
分子量 | 355.43 |
分子式 | C21H25NO4 |
CAS No. | 483-14-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 55 mg/mL (154.74 mM)
H2O: < 1 mg/mL (insoluble or slightly soluble)
Ethanol: < 1 mg/mL (insoluble or slightly soluble)
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Rotundine 483-14-7 GPCR/G Protein Neuroscience Dopamine Receptor 5-HT Receptor 5-hydroxytryptamine Receptor Inhibitor Gindarine Tetrahydropalmatine L-Tetrahydropalmatine Caseanine inhibit Serotonin Receptor (-)-Tetrahydropalmatine inhibitor