store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Dimethindene (Dimetindeno) is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits antihistamine and anticholinergic effects.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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1 mg | 在庫あり | ¥ 45,000 | |||
2 mg | 在庫あり | ¥ 67,500 | |||
5 mg | 在庫あり | ¥ 103,000 | |||
10 mg | 在庫あり | ¥ 151,500 | |||
25 mg | 在庫あり | ¥ 226,500 | |||
50 mg | 在庫あり | ¥ 319,000 | |||
100 mg | 在庫あり | ¥ 431,500 |
説明 | Dimethindene (Dimetindeno) is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits antihistamine and anticholinergic effects. |
In vitro | In follicle-enclosed Xenopus oocytes, Dimethindene (5-500 μM) decreases Cromakalim cromakalim-induced K+ currents (IC50 = 29.5 μM)[1]. |
In vivo | In C57BL/6 mice with skin wound healing, Dimethindene (0.25 mg; i.p.) impairs cutaneous wound healing and delays skin wound closure[2]. |
別名 | Dimetindeno, Z 2001, Dimetindene, Z-2001, Z2001 |
分子量 | 292.42 |
分子式 | C20H24N2 |
CAS No. | 5636-83-9 |
store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Dimethindene 5636-83-9 GPCR/G Protein Immunology/Inflammation Membrane transporter/Ion channel Metabolism Neuroscience Histamine Receptor AChR Endogenous Metabolite Potassium Channel Dimetindeno Z 2001 Dimetindene Z-2001 Z2001 Inhibitor inhibitor inhibit