Powder: -20°C for 3 years | In solvent: -80°C for 1 year
EPZ011989 is a effective, specific orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 Y646 and EZH2 wt; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
2 mg | 在庫あり | ¥ 8,000 | |||
5 mg | 在庫あり | ¥ 12,000 | |||
10 mg | 在庫あり | ¥ 17,500 | |||
25 mg | 在庫あり | ¥ 30,500 | |||
50 mg | 在庫あり | ¥ 49,000 | |||
100 mg | 在庫あり | ¥ 88,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 16,500 |
説明 | EPZ011989 is a effective, specific orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 Y646 and EZH2 wt; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase. |
ターゲット&IC50 | EZH2:<3 nM(Ki), EZH1:103 nM |
分子量 | 605.81 |
分子式 | C35H51N5O4 |
CAS No. | 1598383-40-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 1mg/ml
Ethanol: 100 mg/mL (155.7 mM)
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
EPZ011989 1598383-40-4 Chromatin/Epigenetic Histone Methyltransferase inhibit Inhibitor EPZ 011989 EPZ-011989 inhibitor