Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM, respectively).
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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2 mg | 在庫あり | ¥ 7,500 | |||
5 mg | 在庫あり | ¥ 12,000 | |||
10 mg | 在庫あり | ¥ 20,500 | |||
25 mg | 在庫あり | ¥ 41,000 | |||
50 mg | 在庫あり | ¥ 75,500 | |||
100 mg | 在庫あり | ¥ 112,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 13,000 |
説明 | Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM, respectively). |
ターゲット&IC50 | 5-HT1A:40 nM , 5-HT2B:81 nM, 5-HT1B:52 nM |
In vivo | Eltoprazine hydrochloride exerts a dose-dependent decrease in aggressive behavior in resident-intruder tests with rats (ID50 = 0.24 mg/kg)[1]. |
別名 | DU 28853 hydrochloride |
分子量 | 256.73 |
分子式 | C12H17ClN2O2 |
CAS No. | 98206-09-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 31 mg/mL (120.75 mM)
H2O: 28 mg/mL (109.06 mM)
You can also refer to dose conversion for different animals. 詳細
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Eltoprazine hydrochloride 98206-09-8 GPCR/G Protein Neuroscience 5-HT Receptor DU-28853 DU 28853 Hydrochloride 5-hydroxytryptamine Receptor Inhibitor DU-28853 Hydrochloride DU 28853 DU28853 inhibit Eltoprazine Hydrochloride DU28853 Hydrochloride Serotonin Receptor DU 28853 hydrochloride Eltoprazine inhibitor