Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Glycopyrrolate (Glycopyrrolate bromide) is a muscarinic antagonist used as an antispasmodic, in some disorders of the gastrointestinal tract, and to reduce salivation with some anesthetics.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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5 mg | 在庫あり | ¥ 7,500 | |||
10 mg | 在庫あり | ¥ 11,000 | |||
25 mg | 在庫あり | ¥ 13,500 | |||
50 mg | 在庫あり | ¥ 21,000 | |||
100 mg | 在庫あり | ¥ 30,000 | |||
500 mg | 在庫あり | ¥ 73,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 11,500 |
説明 | Glycopyrrolate (Glycopyrrolate bromide) is a muscarinic antagonist used as an antispasmodic, in some disorders of the gastrointestinal tract, and to reduce salivation with some anesthetics. |
In vitro | Glycopyrrolate inhibits EFS-induced contraction of guinea-pig trachea and human airways in a concentration-dependent manner. In competition studies, glycopyrrolate binds human peripheral lung and human airway smooth muscle (HASM) muscarinic receptors with affinities in the nanomolar range (Ki values 0.5–3.6?nM). Glycopyrrolate showed no selectivity in its binding to the M1–M3 receptors. Kinetics studies show that glycopyrrolate dissociates slowly from HASM muscarinic receptors[1]. |
別名 | Gastrodyn, Glycopyrronium bromide, Robinul, Glycopyrrolate bromide |
分子量 | 398.33 |
分子式 | C19H28BrNO3 |
CAS No. | 596-51-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 60 mg/mL (150.6 mM)
H2O: 72 mg/mL (180.8 mM)
Ethanol: 55 mg/mL (138.1 mM)
You can also refer to dose conversion for different animals. 詳細
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Glycopyrrolate 596-51-0 Neuroscience AChR Glycopyrronium Gastrodyn Glycopyrronium bromide Robinul inhibit Glycopyrrolate Bromide Muscarinic acetylcholine receptor mAChR Glycopyrrolate bromide Inhibitor Glycopyrronium Bromide inhibitor