Powder: -20°C for 3 years | In solvent: -80°C for 1 year
MRS-1706 has Ki values of 1.39, 112, 157, and 230 nM for human A2B, A2A, A1, and A3 receptors respectively. MRS-1706 is an effective and selective adenosine A2B receptor inverse agonist.
説明 | MRS-1706 has Ki values of 1.39, 112, 157, and 230 nM for human A2B, A2A, A1, and A3 receptors respectively. MRS-1706 is an effective and selective adenosine A2B receptor inverse agonist. |
ターゲット&IC50 | A2A receptor (human):112(ki), A3 receptor (human):230 nM, A2 receptor (human):157(ki), A2B receptor (human):(ki)1.39 |
分子量 | 503.55 |
分子式 | C27H29N5O5 |
CAS No. | 264622-53-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 6.4 mg/mL (12.71 mM), Sonication and heating are recommended.
H2O: < 0.1 mg/mL (insoluble)
You can also refer to dose conversion for different animals. 詳細
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