Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Mps1-IN-2 is a potent, selective and ATP-competitive dual Mps1/Plk1 inhibitor.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 7,500 | |||
2 mg | 在庫あり | ¥ 10,500 | |||
5 mg | 在庫あり | ¥ 17,500 | |||
10 mg | 在庫あり | ¥ 33,000 | |||
25 mg | 在庫あり | ¥ 58,500 | |||
50 mg | 在庫あり | ¥ 95,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 19,500 |
説明 | Mps1-IN-2 is a potent, selective and ATP-competitive dual Mps1/Plk1 inhibitor. |
ターゲット&IC50 | Mps1:145 nM |
キナーゼ試験 | mTOR activity is assayed using LanthaScreen Kinase kit reagents. PI(3)K α, β, γ and δ activity are assayed using the PI(3)K HTRF assay kit. The concentration of INK128 necessary to achieve inhibition of enzyme activity by 50% (IC50) is calculated using concentrations ranging from 20 μM to 0.1 nM (12-point curve). IC50?values are determined using a nonlinear regression model. |
分子量 | 480.6 |
分子式 | C26H36N6O3 |
CAS No. | 1228817-38-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 14.3 mg/mL (30 mM)
You can also refer to dose conversion for different animals. 詳細
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Mps1-IN-2 1228817-38-6 Cell Cycle/Checkpoint Cytoskeletal Signaling Kinesin PLK inhibit Inhibitor Monopolar spindle 1 Mps1 Mps1 IN 2 Polo-like Kinase (PLK) Mps1IN2 Mps-1-IN-2 inhibitor