Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PD 117519 (CI947) is an agonist of adenosine receptor
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
2 mg | 在庫あり | ¥ 7,000 | |||
5 mg | 在庫あり | ¥ 11,500 | |||
10 mg | 在庫あり | ¥ 19,000 | |||
25 mg | 在庫あり | ¥ 34,000 | |||
50 mg | 在庫あり | ¥ 62,500 | |||
100 mg | 在庫あり | ¥ 91,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 13,000 |
説明 | PD 117519 (CI947) is an agonist of adenosine receptor |
In vivo | PD 117519?selectively binds to adenosine A2 receptors (IC50 = 30 μM) over A1 receptors (IC50 = 810 μM) in rat brain membranes.?PD 117519 increases heart rate and decreases systolic blood pressure in normotensive dogs when administered at doses of 2 or 10 mg/kg[1]. |
別名 | CI947 |
分子量 | 383.4 |
分子式 | C19H21N5O4 |
CAS No. | 96392-15-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 100 mg/mL (260.82 mM)
You can also refer to dose conversion for different animals. 詳細
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
PD 117519 96392-15-3 GPCR/G Protein Neuroscience Adenosine Receptor CI 947 PD117519 CI-947 Inhibitor P1 receptor PD-117519 CI947 inhibit inhibitor