Powder: -20°C for 3 years | In solvent: -80°C for 1 year
RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 12,500 | |||
5 mg | 在庫あり | ¥ 28,000 | |||
10 mg | 在庫あり | ¥ 48,500 | |||
25 mg | 在庫あり | ¥ 82,000 | |||
50 mg | 在庫あり | ¥ 122,500 | |||
100 mg | 在庫あり | ¥ 176,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 28,000 |
説明 | RG7713 (RO 5028442) has been used in trials studying Autistic Disorder. |
ターゲット&IC50 | V1a receptor (human):1 nM(Ki), V1a receptor (mouse):39nM(Ki) |
In vitro | RO5028442 (compound 8) has excellent binding in and functional affinity for hV1a, moderate mouse affinity, and excellent selectivity versus human V2 (hV2) and human oxytocin (hOT) receptors. RO5028442 shows high solubility. RO5028442 is found to be highly selective against a panel of 89 targets. Finally, RO5028442 is identified as a suitable compound for clinical studies[1]. |
別名 | RO 5028442 |
分子量 | 437.96 |
分子式 | C25H28ClN3O2 |
CAS No. | 920022-47-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 4.38 mg/mL (10 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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RG7713 920022-47-5 GPCR/G Protein Vasopressin Receptor RG-7713 RO 5028442 Inhibitor RG 7713 RO-5028442 RO5028442 inhibit inhibitor