Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Regorafénib N-oxyde M2 is an active metabolite of Regorafenib. Regorafenib is a multi-target inhibitor for VEGFR1/2/3, PDGFRβ, RET, Kit, and Raf-1 (IC50s: 13/4.2/46, 1.5, 22, 7, and 2.5 nM).
説明 | Regorafénib N-oxyde M2 is an active metabolite of Regorafenib. Regorafenib is a multi-target inhibitor for VEGFR1/2/3, PDGFRβ, RET, Kit, and Raf-1 (IC50s: 13/4.2/46, 1.5, 22, 7, and 2.5 nM). |
ターゲット&IC50 | PDGFRβ:1.5nM , c-Kit:7nM , Raf-1:2.5 nM , VEGFR1:13nM , RET:22nM , VEGFR3:46nM , VEGFR2:4.2nM |
分子量 | 498.81 |
分子式 | C21H15ClF4N4O4 |
CAS No. | 835621-11-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: Slightly soluble
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
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