Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, >100 μM and 42 μM for D2 receptor, D1 receptor and α1-adrenoceptor.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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1 mg | 在庫あり | ¥ 18,000 | |||
2 mg | 在庫あり | ¥ 27,500 | |||
5 mg | 在庫あり | ¥ 41,000 | |||
10 mg | 在庫あり | ¥ 49,500 | |||
25 mg | 在庫あり | ¥ 109,000 | |||
50 mg | 在庫あり | ¥ 159,500 | |||
100 mg | 在庫あり | ¥ 227,000 | |||
500 mg | 在庫あり | ¥ 454,500 |
説明 | Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, >100 μM and 42 μM for D2 receptor, D1 receptor and α1-adrenoceptor. |
In vivo | In male Sprague-Dawley rats, Remoxipride hydrochloride (0.1-100 μM/kg; i.p.) blockes apomorphine-induced hyperactivity and dose-dependent blockades apomorphine-induced behaviors. In beagle dogs, Remoxipride hydrochloride (0.25-5 μM/kg; gavage) blockes apomorphine-induced vomiting[1]. |
別名 | Remoxipride Hydrochloride Anhydrous, Roxiam, (S)-Remoxipride Hydrochloride |
分子量 | 407.73 |
分子式 | C16H24BrClN2O3 |
CAS No. | 73220-03-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
H2O: 40.9mg/mL (100mM)
You can also refer to dose conversion for different animals. 詳細
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Remoxipride hydrochloride 73220-03-8 GPCR/G Protein Neuroscience Dopamine Receptor Remoxipride Hydrochloride Anhydrous Roxiam Remoxipride Hydrochloride (S)-Remoxipride Hydrochloride Inhibitor inhibitor inhibit