Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Rotigotine Hydrochloride (N-0924), a dopamine receptor agonist prefering for D3 receptors over D1 and D2, has effective activity of anti-Parkinsonian. Racemic rotigotine hydrochloride is about 50 times as potent as quinpirole, the gold standard D2 agonist.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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サンプルについてお問い合わせ | |||||
5 mg | 在庫あり | ¥ 10,500 | |||
10 mg | 在庫あり | ¥ 15,500 | |||
25 mg | 在庫あり | ¥ 22,500 | |||
50 mg | 在庫あり | ¥ 32,500 | |||
100 mg | 在庫あり | ¥ 45,000 | |||
200 mg | 在庫あり | ¥ 66,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 13,500 |
説明 | Rotigotine Hydrochloride (N-0924), a dopamine receptor agonist prefering for D3 receptors over D1 and D2, has effective activity of anti-Parkinsonian. Racemic rotigotine hydrochloride is about 50 times as potent as quinpirole, the gold standard D2 agonist. |
ターゲット&IC50 | α1B:273 nM (Ki), 5-HT7 receptor:86 nM (Ki), D1 receptor:83 nM (Ki), α2A:338 nM (Ki), D4 receptor:4-15 nM (Ki), D3 receptor:0.71 nM (Ki), 5-HT1A receptor:30 nM (Ki), α2B:27 nM (Ki), D5 receptor:4-15 nM (Ki), D2 receptor:4-15 nM (Ki), α1A:176 nM (Ki) |
別名 | Rotigotine (Hydrochloride), N 0923, N-0924, Rotigotine HCl, N-0923 |
分子量 | 351.93 |
分子式 | C19H26ClNOS |
CAS No. | 125572-93-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (142.07 mM)
You can also refer to dose conversion for different animals. 詳細
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Rotigotine Hydrochloride 125572-93-2 GPCR/G Protein Neuroscience Dopamine Receptor 5-HT Receptor Adrenergic Receptor inhibit Inhibitor Rotigotine (Hydrochloride) N 0924 Rotigotine Serotonin Receptor N 0923 N-0924 Rotigotine HCl Beta Receptor 5-hydroxytryptamine Receptor N0924 N0923 N-0923 inhibitor