Powder: -20°C for 3 years | In solvent: -80°C for 1 year
A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
説明 | A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively. |
ターゲット&IC50 | A2A receptor:4 nM (Ki), A1 receptor:264 nM (Ki) |
In vitro | A2A receptor anyagonist 1 is a potent adenosine A2A receptor antagonist, selective over the A1 receptor and demonstrate its binding activity with Ki values of 4 and 264 nM, respectively. [1] |
別名 | CPI-444 analog, A2A receptor antagonist 1 |
分子量 | 309.3 |
分子式 | C16H12FN5O |
CAS No. | 443103-97-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 20 mg/mL (64.66 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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