Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Compound TPX-0046 is an inhibitor of RET. Compound TPX-0046 can inhibit the RET autophosphorylation. Compound TPX-0046 can be used for the research of cancer.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 49,000 |
5 mg | 在庫あり | ¥ 91,500 |
10 mg | 在庫あり | ¥ 135,500 |
25 mg | 在庫あり | ¥ 217,000 |
50 mg | 在庫あり | ¥ 294,000 |
100 mg | 在庫あり | ¥ 397,000 |
500 mg | 在庫あり | ¥ 794,000 |
説明 | Compound TPX-0046 is an inhibitor of RET. Compound TPX-0046 can inhibit the RET autophosphorylation. Compound TPX-0046 can be used for the research of cancer. |
In vitro | Compound TPX-0046 (0.3-300 nM) inhibits p-RET (y905) in RET-driven cells[1]. |
In vivo | Compound TPX-0046 (2-5 mg/kg; twice daily for 27 days) decreases tumor size in mice[1]. |
分子量 | 424.43 |
分子式 | C21H21FN6O3 |
CAS No. | 2411115-73-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: Slightly soluble
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Compound TPX-0046 2411115-73-4 Apoptosis Tyrosine Kinase/Adaptors c-RET CompoundTPX0046 Compound TPX 0046 Compound TPX0046 Inhibitor inhibitor inhibit