Powder: -20°C for 3 years | In solvent: -80°C for 1 year
IK-930 is an orally active TEAD inhibitor (EC50 < 0.1 µM) with potent potency.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
5 mg | 在庫あり | ¥ 12,000 | |||
10 mg | 在庫あり | ¥ 19,500 | |||
25 mg | 在庫あり | ¥ 39,500 | |||
50 mg | 在庫あり | ¥ 64,000 | |||
100 mg | 在庫あり | ¥ 104,000 |
説明 | IK-930 is an orally active TEAD inhibitor (EC50 < 0.1 µM) with potent potency. |
ターゲット&IC50 | TEAD:<0.1 µM(EC50) |
In vitro | IK-930 (0-1 μM) is a potent and selective TEAD inhibitor.[2] |
In vivo | IK-930 (compound I-32) (10 mg/kg; p.o.) exhibits favorable pharmacokinetic parameters in BALB/c mice with Cmax of 1088 ng/mL and AUC 0-last of 4581 ng*h /mL.[1] |
別名 | compound I-32 |
分子量 | 424.44 |
分子式 | C19H19F3N4O2S |
CAS No. | 2563892-44-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 90.0 mg/mL (212.0 mM), Sonication and heating to 60℃ are recommended.
You can also refer to dose conversion for different animals. 詳細
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
IK-930 2563892-44-2 Stem Cells YAP compound I-32 IK 930 IK930 Inhibitor inhibitor inhibit