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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T6321 | Tofacitinib | Tasocitinib,CP-690550 | ROCK , Apoptosis , JAK , Src |
Tofacitinib (Tasocitinib) is an oral, small molecule inhibitor of Janus kinases that is used to treat moderate-to-severe rheumatoid arthritis. | |||
T13426L | (3S,4S)-Tofacitinib | Others | |
(3S,4S)-Tofacitinib, a less active enantiomer of tofacitinib, is a Janus kinases inhibitor. | |||
T13426 | (3R,4S)-Tofacitinib | Others | |
(3R,4S)-Tofacitinib is an less active enantiomer of Tofacitinib. Tofacitinib is a JAK3 inhibitor(IC50 : 1 nM). | |||
T13427 | (3S,4R)-Tofacitinib | Others | |
(3S,4R)-Tofacitinib is an less active enantiomer of Tofacitinib. Tofacitinib is a JAK3 inhibitor(IC50 : 1 nM). |