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T76566 |
Fsh receptor-binding inhibitor fragment(bi-10)
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FSH receptor-binding inhibitor fragment (bi-10) is a potent antagonist that inhibits the binding of follicle-stimulating hormone (FSH) to its receptor (FSHR), modifying FSH activity at the receptor level. It suppresses o... |
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T1908 |
MHY1485
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mTOR
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Autophagy
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MHY1485 is a mTOR activator. It inhibits the autophagic process by inhibition of fusion between autophagosomes and lysosomes, leading to the accumulation of LC3II protein and enlarged autophagosomes. |
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T3630 |
Relugolix
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RVT-601,TAK-385 |
GNRH Receptor
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Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with potential antineoplastic activity. Relugolix competitively bi... |
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T76222 |
HFSH-β-(33-53) (TFA)
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hFSH-β-(33-53) TFA, a thiol-containing peptide representing the second follicle-stimulating hormone receptor (FSHR) binding domain, acts as an FSHR antagonist. It prevents FSH from binding to its receptor and partially p... |
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T72835 |
FSHR agonist 1
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FSHR agonist 1, an allosteric agonist of the follicle-stimulating hormone receptor (FSHR), exhibits high affinity, with a pEC50 of 7.72. It forms extensive interactions with the transmembrane domain (TMD) to directly act... |
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T9380L |
Antide acetate
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Antide acetate (112568-12-4 Free base) |
LHRH
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Antide acetate is an LHRH antagonist and represses LH and FSH release from the pituitary gland. |
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TP1342L |
GnRH-I acetate
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GnRH-I acetate(33515-09-2 free base) |
Others
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GnRH-I acetate in release of biologically active Follicle-Stimulating Hormone (FSH) and Luteinizing Hormone (LH) in the blood. |
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T5520L |
Cetrorelix diacetate
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NS-75A,SB-075 acetate,SB-075 diacetate,Cetrorelix acetate,NS-75A diacetate |
GNRH Receptor
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Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist. It works by blocking the action of GnRH upon the pituitary, thus rapidly suppressing the production and action of luteinizing hormone (LH) ... |
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T21309 |
Nafarelin acetate(76932-56-4 free base)
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RS-94991-298,Nafarelin acetate,Nafarelin acetate hydrate,Synarel |
GNRH Receptor
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Nafarelin acetate(76932-56-4 free base) (RS-94991-298) is a GnRH agonist that acts as an analog of GnRH. Nafarelin acetate(76932-56-4 free base) causes a decrease in the pituitary secretion of gonadotropins luteinizing h... |
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T2597 |
Norgestrel
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SH-850,FH 122-A,WY-3707,SH-70850 |
Estrogen/progestogen Receptor
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Reactive Oxygen Species
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Norgestrel (WY-3707) is a synthetic progestin commonly used alone or in combination with an estrogen for contraception. Norgestrel suppresses the secretion of luteinizing and follicle-stimulating hormones (LH and FSH), t... |
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T21410 |
Triptorelin acetate(57773-63-4 free base)
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Wy 42422,Triptorelin Acetate,CL 118532,AY 25650,CL 118,532,Wy 42462,BIM 21003 |
GNRH Receptor
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Triptorelin acetate(57773-63-4 free base) (CL 118,532) is used as a GnRH agonist. It decreases pituitary secretion of gonadotropins luteinizing hormone (LH) and follicle-stimulating hormone (FSH) by causing constant stim... |
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T25443 |
FW 34569
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FW-34-569,FW34569,FW 34-569,FW-34569,FW34-569 |
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FW 34569 is an enkephalin analogue. It stimulated growth hormones and prolactin release and inhibited the release of cortisol and LH, while FSH remained unchanged. |
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T83489 |
[Lys8] LH-RH
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[Lys8] LH-RH, an analogue of LH-RH, effectively stimulates the release of luteinizing hormone (LH) and follicle-stimulating hormone (FSH) [1]. |
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T82162 |
Human follicular gonadotropin releasing peptide
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hF-GRP |
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Human Follicular Gonadotropin Releasing Peptide (hF-GRP) is a hormonal peptide that, in vitro, can induce the secretion of pituitary luteinizing hormone (LH) and follicle-stimulating hormone (FSH) [1] [2]. |
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T82307 |
Glp-His-Pro-Gly-NH2
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pGlu-His-Pro-Gly-NH2 |
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pGlu-His-Pro-Gly-NH2, also known as Glp-His-Pro-Gly-NH2, is a tetrapeptide that promotes the release of gonadotropin, luteinizing hormone (LH), and follicle-stimulating hormone (FSH) [1] [2]. |
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T78515 |
Follicle-stimulating hormone
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Others
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Follicle-stimulating hormone (FSH), a heterodimeric glycoprotein synthesized by gonadotrophs in the anterior pituitary gland, influences animal fertility and reproductive performance [1] [2]. |
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T83498 |
[D-Phe2,D-Ala6]-LH-RH
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Wy 18185 |
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[D-Phe2,D-Ala6]-LH-RH is a potent luteinizing hormone-releasing hormone (LH-RH) antagonist with demonstrated activities against LH/FSH-RH and an ability to inhibit ovulation [1]. |
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T70309 |
Dicetrorelix pamoate
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Dicetrorelix pamoate is a synthetic decapeptide with gonadotropin-releasing hormone (GnRH) antagonistic activity. GnRH induces the production and release of luteinizing hormone (LH) and follicle stimulating hormone (FSH)... |
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T21375 |
Clomifene
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Omifin,D,Chloramiphene,Clomiphene,Clomiphene free base,Citrate |
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Clomifene is a selective estrogen receptor modulator (SERM), it has both estrogenic and anti-estrogenic activities. This agent causes the release of the pituitary gonadotropins follicle-stimulating hormone (FSH) and lute... |
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T76620 |
(D-Tyr5,D-Ser(tBu)6,Azagly10)-LHRH
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(D-Tyr5,D-Ser(tBu)6,Azagly10)-LHRH, an analogue of luteinizing hormone-releasing hormone (LHRH), plays a pivotal role in reproductive control by promoting the pituitary release of luteinizing hormone (LH) and follicle-st... |
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T76615 |
(D-Ser(tBu)6,D-Leu7,Azagly10)-LHRH
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(D-Ser(tBu)6,D-Leu7,Azagly10)-LHRH, an analogue of the luteinizing hormone-releasing hormone (LHRH), fundamentally mediates reproductive processes by promoting the secretion of pituitary luteinizing hormone (LH) and foll... |
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T81390 |
Prolactin-Releasing Peptide (1-31) (rat)
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Prolactin-Releasing Peptide (1-31) (rat) serves as a ligand for the UHR-1/GRP10 receptor, moderating fasting-induced food intake and elevating plasma concentrations of LH, FSH, and testosterone in rats [1] [2]. |
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T63572 |
Org 43553
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Org 43553 is an orally active low molecular weight (LMW) luteinizing hormone receptor (LH-R) agonist capable of agonizing human LH (EC50: 3.7 nM) and FSH receptors (EC50: 110 nM).Org 43553 can be used for endocrine studi... |
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T76616 |
(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH
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(D-Ser4, D-Ser(tBu)6, Azagly10)-LHRH, an analogue of luteinizing hormone-releasing hormone (LHRH), plays a pivotal role in reproductive regulation by promoting the secretion of pituitary luteinizing hormone (LH) and foll... |
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T68525 |
Nafarelin acetate hydrate
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Nafarelin is a gonadotropin-releasing hormone agonist (GnRH agonist) which acts as an analog of GnRH. Nafarelin increases the release of FSH and LH by the anterior pituitary, which in turn leads to an increase of estroge... |
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T70670 |
TAK-448 TFA
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TAK-448 is an investigational oligopeptide analog of kisspeptin and a potent agonist of the GPR54 receptor. In animals, acute TAK-448 administration stimulates LH/FSH release, whereas continuous sc exposure rapidly down-... |
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T71149 |
Triptorelin pamoate
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Triptorelin, a decapeptide (pGlu-His-Trp-Ser-Tyr-D-Trp-Leu-Arg-Pro-Gly-NH2), is a gonadotropin-releasing hormone agonist (GnRH agonist) used as the acetate or pamoate salts. By causing constant stimulation of the pituita... |
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T76048 |
TAK-683 acetate
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TAK-683 acetate is a nonapeptide metastin analog and a potent full agonist of the KISS1 receptor (KISS1R), exhibiting IC 50 =170 pM and enhanced metabolic stability. This compound shows agonistic activities towards KISS1... |
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T81270 |
Ripafollitropin alfa (bovine)
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Ripafollitropin alfa (bovine) is a fusion protein that combines recombinant follicle-stimulating hormone with chorionic gonadotropin [1]. |
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T76047 |
TAK-683 TFA
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TAK-683 TFA, a potent full KISS1 receptor (KISS1R) agonist with a half-maximal inhibitory concentration (IC50) of 170 pM, exhibits enhanced metabolic stability. As a nonapeptide metastin analog, it demonstrates agonistic... |
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T68292 |
GTX-758
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GTX-758, also known as Capesaris, is a n orally available, nonsteroidal selective estrogen receptor (ER) alpha agonist with potential antineoplastic activity. Upon administration of GTx-758, this agent suppresses the sec... |
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T35794 |
Kisspeptin-54 (human) (trifluoroacetate salt)
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Kisspeptin-54 is a peptide ligand of the orphan G protein-coupled receptor GPR54 (Kis = 1.81 and 1.45 nM for rat and human receptors, respectively).1 It is a 54 amino acid peptide encoded by the metastasis suppressor gen... |
