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Search Results for " Phenothiazine "

ターゲット

43

阻害剤

カタログ番号 製品名 別名 ターゲット
T0776 Phenothiazine ENT 38 Dopamine Receptor , Antibacterial , Antibiotic , Antifungal
Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities. Phenothiazines antagonize the dopamine D2-receptor in the chemoreceptor trigger zone (CTZ)...
T34189 PTZ-256 phenothiazine derivative,PTZ256
PTZ-256 is a phenothiazine derivative with chemical name: 3-(10H-phenothiazin-10-yl)propane-1-amine. PTZ-256 has molecule weight 256, therefore, we call it as PTZ-256.
T9827 Carfenazine Dopamine Receptor
carfenazine targets the Dopamine receptor and is used for schizophrenia research.
TNU0712 3-(2',5'-Disulfophenylimino)-3H-phenothiazine
3-(2',5'-Disulfophenylimino)-3H-phenothiazine is a bio-reagent and a fine chemical.
TNU0675 3-(4’-Carboxyphenyl)imino-3H-phenothiazine
Bio-reagent, fine chemical
T10232 Acetophenazine dimaleate Dopamine Receptor
Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.
T9353 OXOMEMAZINE AChR , Histamine Receptor
Oxomemazine is a phenothiazine-based histamine H1-receptor blocker with pronounced antimuscarinic activity. Oxomemazine is a selective antagonist of mycotoxins M1 receptors, showing high (Ki=84 nM, M1 receptors) and low ...
T7943 Fluphenazine decanoate Dopamine Receptor
Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.
T0642 2-Methoxyphenothiazine Factor Xa
2-Methoxy Phenothiazine is light yellow or light gray solid.
T0622 2-Chlorophenothiazine Others
2-Chlorophenothiazine is used as the intermediate of Chlorpromazine hydrochloride.
T4117 Zuclopenthixol cis-Clopenthixol,Cisordinol,(Z)-Clopenthixol Dopamine Receptor
Zuclopenthixol (cis-Clopenthixol) is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors.
T0385 Prochlorperazine Maleate Prochlorperazin,Capazine,Prochlorperazine dimaleate salt,Stemetil,Compazine Dopamine Receptor
Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO. It is more likely than CHLORPROMAZINE to cause EXTRAPYRAMIDAL DISORDERS.
T12777 RTC-5 TRC-382 EGFR
RTC-5 (TRC-382) is a phenothiazine compound that has been specifically enhanced for its potent anti-cancer properties. It exhibits considerable effectiveness against an EGFR-driven cancer xenograft model. The mechanism ...
T0068 Fluphenazine dihydrochloride Prolixin,Fluphenazine hydrochloride Dopamine Receptor
Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR; In studies, Fluphenazine can be used to probe the effects and metabolic process of this commonly used dopamine antagonist.
T0766 Promazine hydrochloride Romtiazin hydrochloride,Sinophenin hydrochloride Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , AChR
Promazine hydrochloride (Romtiazin hydrochloride) is a phenothiazine with actions similar to CHLORPROMAZINE but with less antipsychotic activity. It is primarily used in short-term treatment of disturbed behavior and as ...
T1090 Perphenazine Perphenazin,Etaperazine,Trilafon CaMK , Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
T50054 Opromazine hydrochloride Others
Opromazine hydrochloride belongs to the phenothiazine class of antipsychotics and reduces the activity of dopaminergic pathways by blocking dopamine receptors in the brain. It is mainly used for the treatment of psychiat...
T0312 Toluidine Blue Blutene chloride Others
Toluidine Blue (Blutene chloride), a phenothiazine, is used as a biological stain, a hemostatic, and a dye for silk and wool. Blutene chloride is also used as a diagnostic aid for gastric neoplasms and oral, and used in ...
T0302L Triflupromazine Vesprin,Fluopromazine,Trifluopromazine,Adazine,Siquil
Triflupromazine is a phenothiazine drug used as an antipsychotic and antiemetic.
T23843L Butaperazine maleate Tyrylen,Repoise maleate
Butaperazine maleate, a phenothiazine derivative, is an antipsychotic.
T23843 Butaperazine Butyrylyperazine,Bayer 1362,Butaperazina,Butyrylperazine
Butaperazine is a typical antipsychotic of the phenothiazine class.
T40854 Imiclopazine
Imiclopazine is a phenothiazine derivative with good sedative, analgesic, antiaggressive and antiemetic effects.
T33319 Methdilazine Hydrochloride Bristaline,Dilosyn,Methdilazine Hcl,Tacaryl hydrochloride,Disyncran
Methdilazine Hydrochloride is a first-generation phenothiazine class antihistamine with anticholinergic properties.
T19525 PPA-904 Others
PPA-904 is a specific phenothiazine photosensitizer,and used in photodynamic therapy.
T0445L1 Promethazine hibenzate D-08768,D08768,D 08768
Promethazine is a neuroleptic medication and first-generation antihistamine of the phenothiazine family.
T69407 Fonazine hydrochloride
Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.
T70997 Fonazine mesylate
Fonazine mesylate is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.
T31844 Fonazine Dimethodin,Banistyl,Dimetiotazine,Dimetotiazine,Dimethothiazine
Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.
T15026 Cyamemazine 5-HT Receptor
Cyamemazine, contains the phenothiazine chromophore, is a neuroleptic agent used as an anxiolytic. Cyamemazine is a potent 5-HT3 (Ki: 12 nM), 5-HT2A (Ki: 1.5 nM) and 5-HT2C (Ki: 75 nM) receptors antagonist with antipsych...
T71160 Levomepromazine HCl
Levomepromazine HCl is a phenothiazine with pharmacological activity similar to that of both CHLORPROMAZINE and PROMETHAZINE. It has the histamine-antagonist properties of the antihistamines together with CENTRAL NERVOUS...
T3086L Mesoridazine free base NSC-186066,NSC 186066,NSC186066,TPS23,Mesoridazine,NC-123
Mesoridazine (thioridazine EP impurity B) is a phenothiazine antipsychotic with effects similar to chlorpromazine.
T81348 PTZ-LD
PTZ-LD, a phenothiazine-based fluorescent probe, specifically detects lipid droplets (LDs) with apparent emissivity (Ex/Em=488/570-620 nm) and is utilized in diabetic cataract (DC) research [1].
T31169 D54 naponate
D54 Naponate is a stored salt form of biologically active phenothiazine, which has good antitumor activity and can be maintained longer in the body.
T23949 Dacemazine hydrochloride Ahistan HCl,Dacemazine HCl,Histantine HCl,UNII-DK78VKA001
Dacemazine is a phenothiazine derivative that acts as a histamine antagonist at the H1 subtype. It was also assessed as a possible anticancer drug.
T68193 Clopenthixol
Clopenthixol is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors.
T69103 Clopenthixol decanoate
Clopenthixol decanoate is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors.
T68963 Alpha-Clopenthixol dihydrochloride
alpha-Clopenthixol dihydrochloride is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors.
T18652 RTC-30 Others
RTC-30 is an optimized phenothiazine compound possessing potent anti-cancer properties. It is formulated with a hydroxylated linker (N) which enhances its oral bioavailability[1].
T28282 Oxypertine Win-18501,Forit,Win18501,Win 18501
Oxypertine is an indole-derivative antipsychotic with general properties similar to those of the chlorpromazine and phenothiazine. Oxypertine is used as a treatment for various psychoses including mania, schizophrenia, ...
T68133 Quisultazine
Quisultazine is a phenothiazine derivative with no central effects, can be classified as a non anti H2 antisecretory agent.
T34072 Pipotiazine 19366 RP,Pipotiazina,Pipotiazinum,Piportil L4,Pipothiazine
Pipotiazine has less sedating and a weak propensity for causing hypotension or potentiating the effects of CNS depressants and anesthetics among the different phenothiazine derivatives. However, it produces a high incide...
T0218 Biperiden Bipariden,Akineton,KL 373,Biperidine AChR
Biperiden (Bipariden) is a muscarinic antagonist that has effects in both the central and peripheral nervous systems. It has been used in the treatment of arteriosclerotic, idiopathic, and postencephalitic parkinsonism. ...
T61915 Thiethylperazine
Thiethylperazine is a phenothiazine derivative. Thiethylperazine is a histamine H1 receptor and dopamine D2 receptor antagonist with oral activity. Thiethylperazine is also a selective ABCC1 activator, which can reduce a...

Compounds

Phenothiazine
T0776
Synonym: ENT 38
Target: Dopamine Receptor, Antibacterial, Antibiotic, Antifungal
PTZ-256
T34189
Synonym: phenothiazine derivative,PTZ256
Target:
carfenazine
T9827
Synonym:
Target: Dopamine Receptor
3-(2',5'-Disulfophenylimino)-3H-phenothiazine
TNU0712
Synonym:
Target:
3-(4’-Carboxyphenyl)imino-3H-phenothiazine
TNU0675
Synonym:
Target:
Acetophenazine dimaleate
T10232
Synonym:
Target: Dopamine Receptor
OXOMEMAZINE
T9353
Synonym:
Target: AChR, Histamine Receptor
Fluphenazine decanoate
T7943
Synonym:
Target: Dopamine Receptor
2-Methoxyphenothiazine
T0642
Synonym:
Target: Factor Xa
2-Chlorophenothiazine
T0622
Synonym:
Target: Others
Zuclopenthixol
T4117
Synonym: cis-Clopenthixol,Cisordinol,(Z)-Clopenthixol
Target: Dopamine Receptor
Prochlorperazine Maleate
T0385
Synonym: Prochlorperazin,Capazine,Prochlorperazine dimaleate salt,Stemetil,Compazine
Target: Dopamine Receptor
RTC-5
T12777
Synonym: TRC-382
Target: EGFR
Fluphenazine dihydrochloride
T0068
Synonym: Prolixin,Fluphenazine hydrochloride
Target: Dopamine Receptor
Promazine hydrochloride
T0766
Synonym: Romtiazin hydrochloride,Sinophenin hydrochloride
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, AChR
Perphenazine
T1090
Synonym: Perphenazin,Etaperazine,Trilafon
Target: CaMK, Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
Opromazine hydrochloride
T50054
Synonym:
Target: Others
Toluidine Blue
T0312
Synonym: Blutene chloride
Target: Others
Triflupromazine
T0302L
Synonym: Vesprin,Fluopromazine,Trifluopromazine,Adazine,Siquil
Target:
Butaperazine maleate
T23843L
Synonym: Tyrylen,Repoise maleate
Target:
Butaperazine
T23843
Synonym: Butyrylyperazine,Bayer 1362,Butaperazina,Butyrylperazine
Target:
Imiclopazine
T40854
Synonym:
Target:
Methdilazine Hydrochloride
T33319
Synonym: Bristaline,Dilosyn,Methdilazine Hcl,Tacaryl hydrochloride,Disyncran
Target:
PPA-904
T19525
Synonym:
Target: Others
Promethazine hibenzate
T0445L1
Synonym: D-08768,D08768,D 08768
Target:
Fonazine hydrochloride
T69407
Synonym:
Target:
Fonazine mesylate
T70997
Synonym:
Target:
Fonazine
T31844
Synonym: Dimethodin,Banistyl,Dimetiotazine,Dimetotiazine,Dimethothiazine
Target:
Cyamemazine
T15026
Synonym:
Target: 5-HT Receptor
Levomepromazine HCl
T71160
Synonym:
Target:
Mesoridazine free base
T3086L
Synonym: NSC-186066,NSC 186066,NSC186066,TPS23,Mesoridazine,NC-123
Target:
PTZ-LD
T81348
Synonym:
Target:
D54 naponate
T31169
Synonym:
Target:
Dacemazine hydrochloride
T23949
Synonym: Ahistan HCl,Dacemazine HCl,Histantine HCl,UNII-DK78VKA001
Target:
Clopenthixol
T68193
Synonym:
Target:
Clopenthixol decanoate
T69103
Synonym:
Target:
alpha-Clopenthixol dihydrochloride
T68963
Synonym:
Target:
RTC-30
T18652
Synonym:
Target: Others
Oxypertine
T28282
Synonym: Win-18501,Forit,Win18501,Win 18501
Target:
quisultazine
T68133
Synonym:
Target:
Pipotiazine
T34072
Synonym: 19366 RP,Pipotiazina,Pipotiazinum,Piportil L4,Pipothiazine
Target:
Biperiden
T0218
Synonym: Bipariden,Akineton,KL 373,Biperidine
Target: AChR
Thiethylperazine
T61915
Synonym:
Target: