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カタログ番号 | 製品名 | 別名 | ターゲット |
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T0776 | Phenothiazine | ENT 38 | Dopamine Receptor , Antibacterial , Antibiotic , Antifungal |
Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities. Phenothiazines antagonize the dopamine D2-receptor in the chemoreceptor trigger zone (CTZ)... | |||
T34189 | PTZ-256 | phenothiazine derivative,PTZ256 | |
PTZ-256 is a phenothiazine derivative with chemical name: 3-(10H-phenothiazin-10-yl)propane-1-amine. PTZ-256 has molecule weight 256, therefore, we call it as PTZ-256. | |||
T9827 | Carfenazine | Dopamine Receptor | |
carfenazine targets the Dopamine receptor and is used for schizophrenia research. | |||
TNU0675 | 3-(4’-Carboxyphenyl)imino-3H-phenothiazine | ||
3-(4'-Carboxyphenyl)imino-3H-phenothiazine is a Bio-reagent, fine chemical. | |||
TNU0712 | 3-(2',5'-Disulfophenylimino)-3H-phenothiazine | ||
3-(2',5'-Disulfophenylimino)-3H-phenothiazine is a Bio-reagent, fine chemical. | |||
T10232 | Acetophenazine dimaleate | Dopamine Receptor | |
Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor. | |||
T9353 | OXOMEMAZINE | AChR , Histamine Receptor | |
Oxomemazine is a phenothiazine-based histamine H1-receptor blocker with pronounced antimuscarinic activity. Oxomemazine is a selective antagonist of mycotoxins M1 receptors, showing high (Ki=84 nM, M1 receptors) and low ... | |||
T7943 | Fluphenazine decanoate | Dopamine Receptor | |
Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia. | |||
T0642 | 2-Methoxyphenothiazine | Factor Xa | |
2-Methoxy Phenothiazine is light yellow or light gray solid. | |||
T0622 | 2-Chlorophenothiazine | Others | |
2-Chlorophenothiazine is used as the intermediate of Chlorpromazine hydrochloride. | |||
T4117 | Zuclopenthixol | cis-Clopenthixol,Cisordinol,(Z)-Clopenthixol | Dopamine Receptor |
Zuclopenthixol (cis-Clopenthixol) is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors. | |||
T12777 | RTC-5 | TRC-382 | EGFR |
RTC-5 (TRC-382) is a phenothiazine compound that has been specifically enhanced for its potent anti-cancer properties. It exhibits considerable effectiveness against an EGFR-driven cancer xenograft model. The mechanism ... | |||
T0385 | Prochlorperazine Maleate | Prochlorperazin,Capazine,Prochlorperazine dimaleate salt,Stemetil,Compazine | Dopamine Receptor |
Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO. It is more likely than CHLORPROMAZINE to cause EXTRAPYRAMIDAL DISORDERS. | |||
T0068 | Fluphenazine dihydrochloride | Prolixin,Fluphenazine hydrochloride | Dopamine Receptor |
Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR; In studies, Fluphenazine can be used to probe the effects and metabolic process of this commonly used dopamine antagonist. | |||
T0766 | Promazine hydrochloride | Romtiazin hydrochloride,Sinophenin hydrochloride | Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , AChR |
Promazine hydrochloride (Romtiazin hydrochloride) is a phenothiazine with actions similar to CHLORPROMAZINE but with less antipsychotic activity. It is primarily used in short-term treatment of disturbed behavior and as ... | |||
T1090 | Perphenazine | Perphenazin,Etaperazine,Trilafon | CaMK , Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Histamine Receptor |
Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties. | |||
T50054 | Opromazine hydrochloride | Others | |
Opromazine hydrochloride belongs to the phenothiazine class of antipsychotics and reduces the activity of dopaminergic pathways by blocking dopamine receptors in the brain. It is mainly used for the treatment of psychiat... | |||
T0312 | Toluidine Blue | Blutene chloride | Others |
Toluidine Blue (Blutene chloride), a phenothiazine, is used as a biological stain, a hemostatic, and a dye for silk and wool. Blutene chloride is also used as a diagnostic aid for gastric neoplasms and oral, and used in ... | |||
T0302L | Triflupromazine | Vesprin,Fluopromazine,Trifluopromazine,Adazine,Siquil | |
Triflupromazine is a phenothiazine drug used as an antipsychotic and antiemetic. | |||
T40854 | Imiclopazine | ||
Imiclopazine is a phenothiazine derivative with good sedative, analgesic, antiaggressive and antiemetic effects. | |||
T23843L | Butaperazine maleate | Tyrylen,Repoise maleate | |
Butaperazine maleate, a phenothiazine derivative, is an antipsychotic. | |||
T23843 | Butaperazine | Butyrylyperazine,Bayer 1362,Butaperazina,Butyrylperazine | |
Butaperazine is a typical antipsychotic of the phenothiazine class. | |||
T69407 | Fonazine hydrochloride | ||
Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist. | |||
T70997 | Fonazine mesylate | ||
Fonazine mesylate is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist. | |||
T33319 | Methdilazine Hydrochloride | Bristaline,Dilosyn,Methdilazine Hcl,Tacaryl hydrochloride,Disyncran | |
Methdilazine Hydrochloride is a first-generation phenothiazine class antihistamine with anticholinergic properties. | |||
T19525 | PPA-904 | Others | |
PPA-904 is a specific phenothiazine photosensitizer,and used in photodynamic therapy. | |||
T0445L1 | Promethazine hibenzate | D-08768,D08768,D 08768 | |
Promethazine is a neuroleptic medication and first-generation antihistamine of the phenothiazine family. | |||
T15026 | Cyamemazine | 5-HT Receptor | |
Cyamemazine, contains the phenothiazine chromophore, is a neuroleptic agent used as an anxiolytic. Cyamemazine is a potent 5-HT3 (Ki: 12 nM), 5-HT2A (Ki: 1.5 nM) and 5-HT2C (Ki: 75 nM) receptors antagonist with antipsych... | |||
T31844 | Fonazine | Dimethodin,Banistyl,Dimetiotazine,Dimetotiazine,Dimethothiazine | |
Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist. | |||
T71160 | Levomepromazine HCl | ||
Levomepromazine HCl is a phenothiazine with pharmacological activity similar to that of both CHLORPROMAZINE and PROMETHAZINE. It has the histamine-antagonist properties of the antihistamines together with CENTRAL NERVOUS... | |||
T3086L | Mesoridazine free base | NSC-186066,NSC 186066,NSC186066,TPS23,Mesoridazine,NC-123 | |
Mesoridazine (thioridazine EP impurity B) is a phenothiazine antipsychotic with effects similar to chlorpromazine. | |||
T81348 | PTZ-LD | ||
PTZ-LD, a phenothiazine-based fluorescent probe, specifically detects lipid droplets (LDs) with apparent emissivity (Ex/Em=488/570-620 nm) and is utilized in diabetic cataract (DC) research [1]. | |||
T31169 | D54 naponate | ||
D54 Naponate is a stored salt form of biologically active phenothiazine, which has good antitumor activity and can be maintained longer in the body. | |||
T23949 | Dacemazine hydrochloride | Ahistan HCl,Dacemazine HCl,Histantine HCl,UNII-DK78VKA001 | |
Dacemazine is a phenothiazine derivative that acts as a histamine antagonist at the H1 subtype. It was also assessed as a possible anticancer drug. | |||
T68193 | Clopenthixol | ||
Clopenthixol is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors. | |||
T69103 | Clopenthixol decanoate | ||
Clopenthixol decanoate is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors. | |||
T68963 | Alpha-Clopenthixol dihydrochloride | ||
alpha-Clopenthixol dihydrochloride is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors. | |||
T18652 | RTC-30 | Others | |
RTC-30 is an optimized phenothiazine compound possessing potent anti-cancer properties. It is formulated with a hydroxylated linker (N) which enhances its oral bioavailability[1]. | |||
T28282 | Oxypertine | Win-18501,Forit,Win18501,Win 18501 | |
Oxypertine is an indole-derivative antipsychotic with general properties similar to those of the chlorpromazine and phenothiazine. Oxypertine is used as a treatment for various psychoses including mania, schizophrenia, ... | |||
T34072 | Pipotiazine | 19366 RP,Pipotiazina,Pipotiazinum,Piportil L4,Pipothiazine | |
Pipotiazine has less sedating and a weak propensity for causing hypotension or potentiating the effects of CNS depressants and anesthetics among the different phenothiazine derivatives. However, it produces a high incide... | |||
T68133 | Quisultazine | ||
Quisultazine is a phenothiazine derivative with no central effects, can be classified as a non anti H2 antisecretory agent. | |||
T0218 | Biperiden | Bipariden,Akineton,KL 373,Biperidine | AChR |
Biperiden (Bipariden) is a muscarinic antagonist that has effects in both the central and peripheral nervous systems. It has been used in the treatment of arteriosclerotic, idiopathic, and postencephalitic parkinsonism. ... | |||
T61915 | Thiethylperazine | ||
Thiethylperazine is a phenothiazine derivative. Thiethylperazine is a histamine H1 receptor and dopamine D2 receptor antagonist with oral activity. Thiethylperazine is also a selective ABCC1 activator, which can reduce a... |