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T13920L |
Terlipressin Acetate
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Terlipressin diacetate anhydrous,Terlipressin acetate anhydrous |
Vasopressin Receptor
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Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on oxygen and glucose deprivation/re-oxygenation (OGD/R)-induced damage in intestinal epithelial cells (IEC-6).Terlipressin acetate exerts anti-in... |
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T2568 |
Felypressin
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Octapressin,Felypressin Acetate,PLV-2,H-[Cys-Phe-Phe-Gln-Asn-Cys]-Pro-Lys-Gly-NH2 |
Vasopressin Receptor
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Felypressin (Octapressin) is a synthetic analog of LYPRESSIN with a PHENYLALANINE substitution at residue 2. Felypressin is a vasoconstrictor with reduced antidiuretic activity. |
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T2568L |
Felypressin acetate
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2-(L-Phenylalanine)-8-L-lysinevasopressin,PLV2. H-Cys-Phe-Phe-Gln-Asn-Cys-Pro-Lys-Gly-NH2 (Disulfide bond),PLV 2,PLV-2 |
Vasopressin Receptor
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Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS. Felypressin acetate can be used in dental procedures. |
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TP1049L |
Ornipressin Acetate（3397-23-7，free）
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Orpressin,POR-8 |
Others
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Ornipressin Acetate (POR-8) is a potent vasoconstrictor, hemostatic and renal agent. |
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T21708L |
Angiotensin 1/2 + A (2 - 8) Acetate
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Angiotensin 1/2 + A (2 - 8) Acetate (51833-76-2 Free base) |
Others
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Angiotensin 1/2 + A (2 - 8) Acetate is a Vasoconstrictor. |
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T0446 |
Naphazoline hydrochloride
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Albalon,Rhinantin,Naphazoline HCl |
Adrenergic Receptor
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Naphazoline hydrochloride (Naphazoline HCl) is an adrenergic vasoconstrictor agent used as a decongestant. |
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T0045 |
Heptaminol hydrochloride
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RP-2831 hydrochloride |
Others
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Heptaminol hydrochloride (RP-2831 hydrochloride), a vasoconstrictor, is used in the therapy of hypotension, especially orthostatic hypotension. |
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TP1737L |
Urotensin II (114-124), human acetate
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Urotensin II (114-124), human acetate(251293-28-4 free base) |
GPR
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Urotensin II (114-124), human acetate is an 11-amino acid residue peptide, is a potent vasoconstrictor and agonist for the orphan receptor GPR14. |
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T7386 |
Bretylium tosylate
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Others
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Bretylium tosylate is an inhibitor of the presynaptic release of vasoconstrictor neurotransmitters, a available antiarrhythmic drug for ventricular arrhythmias. |
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T21445 |
Naphazoline
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AK-Con,Naphcon-a,Clear Eyes,All Clear |
Adrenergic Receptor
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Naphazoline (Naphcon-a) is a sympathomimetic compound with marked alpha adrenergic activity. Naphazoline can be used as a vasoconstrictor with a rapid action in reducing swelling when applied to mucous membrane. |
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TP2165 |
Urotensin II, mouse acetate (9047-55-6 free base)
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Urotensin II, mouse acetate |
GPR
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Urotensin II, mouse acetate (9047-55-6 free base) is an endogenous ligand for the orphan GPR14 or SENR. It is a potent vasoconstrictor. |
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T12924 |
Sitaxsentan
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TBC-11251,IPI 1040 |
Endothelin Receptor
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Sitaxsentan (TBC-11251) is A selective endothelin A (ETA) receptor antagonist. Endothelin is an effective vasoconstrictor. Sitaxsentan blocks the binding of endothelin to its receptors, thereby eliminating the harmful ef... |
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T14021 |
20-HETE
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20-hydroxy Arachidonic Acid |
Others
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20-HETE (20-hydroxy Arachidonic Acid) is a CYP450 metabolite and a potent vasoconstrictor and it is an endogenous inhibitor of the large-conductance Ca2+-activated K+ channel in renal arterioles. 20-HETE increases NADPH ... |
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TP1295 |
Angiotensin I (human, mouse, rat)
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Angiotensin 1 Human |
Others
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Angiotensin I (human, mouse, rat) is the precursor to the vasoconstrictor peptide angiotensin II, cleaved by the angiotensin-converting enzyme (ACE).Angiotensin is a peptide hormone that causes vasoconstriction and an in... |
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T0279 |
Metaraminol tartrate
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Metaradrine tartrate,Metaraminol bitartrate |
Adrenergic Receptor
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Metaraminol tartrate (Metaradrine tartrate) is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors. It has been used primarily as a vasoconstrictor in the treatment of HYPOTENSION. |
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T1462 |
Captopril
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SQ 14225,SQ-14534,SA333 |
RAAS
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Captopril (SA333) is a potent and specific inhibitor of peptidyl-dipeptidase A. It blocks the conversion of angiotensin I to angiotensin II, a vasoconstrictor and important regulator of arterial blood pressure. |
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T19309L1 |
Endothelin 1 (swine, human) acetate
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Endothelin 1 (swine, human) acetate(117399-94-7 free base) |
Endothelin Receptor
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Endothelin 1 (swine, human) acetate is a synthetic peptide with the sequence of human and swine Endothelin 1. Endothelin 1 is a potent endogenous vasoconstrictor and acts through two types of receptors ETA and ETB. |
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T0948 |
Adrenalone hydrochloride
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Adrenalone HCl |
Adrenergic Receptor
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Adrenalone hydrochloride (Adrenalone HCl) is a dopamine β-oxidase inhibitor with a similar structure to the norepinephrine transporter (NET) ligand, with an IC50 of 36.9 μM. It is an adrenergic agonist that acts as a loc... |
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T8560 |
Angiotensin II human acetate
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Ang II acetate,DRVYIHPF acetate,Angiotensin II acetate |
Apoptosis
,
RAAS
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Angiotensin II human acetate (DRVYIHPF acetate) is a vasoconstrictor that mainly acts on the AT1 receptor. |
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TP1345 |
Kisspeptin-10, human (TFA)(374675-21-5,FREE)
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GPR
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Kisspeptin
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Kisspeptin-10, human TFA is a potent vasoconstrictor and angiogenesis inhibitor. Kisspeptin-10, human TFA acts as a tumor metastasis suppressor via its receptor GPR54. Kisspeptin-10-GPR54 system plays an important role i... |
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T6264 |
Bosentan
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Actelion,Ro 47-0203,Benzenesulfonamide |
Endothelin Receptor
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Bosentan (Benzenesulfonamide) is a sulfonamide-derived, competitive and specific endothelin receptor antagonist with a slightly higher affinity for the endothelin A receptor than endothelin B receptor. Bosentan blocks th... |
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T6529 |
Halobetasol propionate
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Halobetasol Propionate,Ulobetasol propionate,BMY-30056,CGP-14458 |
Phospholipase
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Halobetasol propionate (BMY-30056) is the propionate salt form of halobetasol, a synthetic corticosteroid with anti-inflammatory, antipruritic, and vasoconstrictor activities. Halobetasol, a topical steroid, diffuses acr... |
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T0871 |
Noradrenaline bitartrate
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Adrenergic Receptor
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Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors. Norepinephrine Bitartrate is a bitartrate salt of norepinephrine, a synthetic phenylethylamine that mimics the sympathomimetic actions of the ... |
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T13920 |
Terlipressin
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Others
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Terlipressin is a potent vasoconstrictor that acts via V1 receptors on arteriolar smooth muscle cells. |
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T24541 |
Norbormide
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Mcneil 1025,S 6999,MCN 1025,Shoxin,Raticate |
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Norbormide is a toxic compound used as a rodenticide. It has several mechanisms of action, acting as a vasoconstrictor and calcium channel blocker. |
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T0279L2 |
Metaraminol hydrochloride
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Metaraminol HCl |
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Metaraminol hydrochloride, used primarily as a vasoconstrictor in the treatment of HYPOTENSION, is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors. |
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T81652 |
Nordefrin
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(±)-Cobefri |
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Nordefrin ((±)-Cobefri), a derivative of Norepinephrine, acts as a vasoconstrictor [1]. |
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T24603 |
PD-34799-SA
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PD 34799-SA,PD34799-SA |
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PD-34799-SA is an effective inhibitor of vasoconstrictor responses to sympathetic nerve stimulation. |
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T19309 |
Endothelin 1 (swine, human)
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Others
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Endothelin 1 (swine, human), a synthetic peptide mirroring the sequence of both human and swine Endothelin 1, functions as a robust endogenous vasoconstrictor by interacting with two receptor types, ETA and ETB. |
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TP1175 |
Endothelin-3, human, mouse, rabbit, rat
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Endothelin 3 (Rat,Human) |
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Endothelin-3, human, mouse, rabbit, rat , is a cyclic 21 amino acid peptide. It is an endogenous neuropeptide and potent vasoconstrictor. |
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T25199 |
Cafaminol
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Cafaminolum,G1,G-1,G 1 |
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Cafaminol (methylcoffanolamine) is a vasoconstrictor and anticatarrhal of the methylxanthine family related to caffeine which is used as a nasal decongestant. |
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TP1049 |
Ornipressin
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POR-8 |
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Ornipressin is a vasoconstrictor, haemostatic and renal agent. |
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TP1522 |
Angiotensin II (5-8), human
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Angiotensin II (5-8) is an endogenous C-terminal fragment of the peptide vasoconstrictor angiotensin II |
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T69670 |
Clonazoline HCl
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Clonazoline HCl is the salt form of Clonazoline, a coronary vasodilator that is an imidazoline sympathomimetic, an alpha-adrenoreceptor agonist. It was used as a nasal decongestant and vasoconstrictor. |
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T70216 |
Clonazoline
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Clonazoline is a coronary vasodilator that is an imidazoline sympathomimetic, an alpha-adrenoreceptor agonist. It was used as a nasal decongestant and vasoconstrictor. |
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TP1396 |
Kisspeptin-10, human
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Kisspeptin-10, human is an effective vasoconstrictor and inhibitor of angiogenesis. |
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TP1737 |
Urotensin II (114-124), human
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Urotensin II (114-124), human, is an 11-amino acid residue peptide that exhibits strong vasoconstrictor activity and acts as an agonist for the orphan receptor GPR14. |
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T36617 |
Ent-8-iso Prostaglandin F2α
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ent-8-iso Prostaglandin F2α |
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ent-8-iso Prostaglandin F2α is a potent vasoconstrictor of porcine retinal and cerebral microvessels with EC50 values of 30.6 and 53.5 nM, respectively. |
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TP1661 |
Angiotensin II (1-4), human TFA
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Angiotensin II is a potent direct vasoconstrictor, causing arteries and veins to constrict, so leading to an increase in blood pressure. |
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TP1415 |
Urotensin II (114-124), human TFA
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Urotensin II (114-124), human TFA, is an 11-amino acid residue peptide with a strong vasoconstrictor effect. This compound acts as an agonist for the orphan receptor GPR14. |
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T76564 |
Endothelin-1 (1-31) (Human)
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Endothelin-1 (1-31) (Human) is a powerful vasoconstrictor and agent for inducing hypertension, originating from the specific hydrolysis of big ET-1 by chymase [1]. |
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T76564L |
Endothelin-1 (1-31) (Human) acetate
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Endothelin-1 (1-31) (Human) acetate, a potent vasoconstrictor and hypertensive agent, is produced through the selective hydrolysis of big ET-1 by chymase [1]. |
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TP2166 |
Urotensin II, mouse TFA (9047-55-6 free base)
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Urotensin II, mouse TFA |
GPR
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Urotensin II, mouse TFA is an endogenous ligand for the orphan GPR14 or SENR. It is a potent vasoconstrictor. |
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T68825 |
Doxazosin HCl
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Doxazosin HCl is the salt form of Doxazosin Free Base which acts by inhibiting the postsynaptic alpha(1)-adrenoceptors on vascular smooth muscle. This inhibits the vasoconstrictor effect of circulating and locally releas... |
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T78063 |
Endothelin-1 (1-31) (Human) TFA
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ERK
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Endothelin-1 (1-31) (Human) TFA, a potent vasoconstrictor and hypertensive agent, originates from the chymase-mediated selective hydrolysis of big ET-1 [1]. |
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T36479 |
Big Endothelin-1 (1-38), human
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Human Big ET-1 comprises residues 53-90 of the endothelin precursor (preproendothelin). Compared to the mature endothelin-1 (hET-1), the peptide show less vasoconstrictor activity in vitro, but similar pressor effects in... |
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T36480 |
Big Endothelin-1 (1-39), porcine
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The big endothelins comprise residues 53-90 (human big ET-1) and 53-91 (porcine big ET-1) of the endothelin precursor (preproendothelin). Compared to the mature endothelin-1 (ET-1), both peptides show less vasoconstricto... |
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T19631 |
PD 109488
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PD-109488,Quinapril Diketopiperazine,PD109488 |
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PD 109488 is a metabolite of quinapril and is a derivative of Quinapril that acts as an ACE inhibitor. Inhibition of ACE prevents the conversion of signaling peptide angiotensin I into angiotensin II, which acts as a pot... |
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T37227 |
(±)8(9)-DiHET
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Epoxide hydrolases convert the EETs into vicinal diols, with the concurrent loss of much of their biological activity. The 8(S),9(R)-EET isomer is metabolized by platelet COX to form 8(S),9(R),11(R)-THETA, a trihydroxy f... |
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TP1609 |
Angiotensin II (1-4), human
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Angiotensin II is a potent direct vasoconstrictor, causing arteries and veins to constrict, so leading to an increase in blood pressure. Angiotensin also potentiates the release of norepinephrine by a direct action on po... |
