ペプチド
抗体
色素試薬
PROTAC
バーチャルスクリーニング
TargetMolキット
Cell Counting Kit-8 (CCK-8)
Inhibitor Cocktails
天然化合物
フェノール類
アルカロイド類
フラボノイド類
阻害剤
血管新生
アポトーシス
オートファジー
細胞周期・チェックポイント
クロマチン・エピジェネティック
細胞骨格シグナル
DNA損傷・DNA修復
内分泌・ホルモン
GPCR/Gタンパク質
免疫・炎症
JAK・STATシグナル
| Cat. No. | 製品名 | CAS No. | Purity | Chemical Structure |
|---|---|---|---|---|
| T6893 | MK-886 | 118414-82-7 | 98% |
|
| MK-886 is an inhibitor of leukotriene biosynthesis, inhibiting 5-lipoxygenase-activating protein (FLAP). It is also a moderately potent PPARα antagonist. | ||||
| T12835 | Saroglitazar | 495399-09-2 | 98% |
|
| Saroglitazar is an agonist of PPAR with EC50 values of 0.65 pM and 3 nM for PPARα and PPARγ. | ||||
| T6829 | EPI-001 | 227947-06-0 | 98% |
|
| EPI-001 is an androgen receptor N-terminal domain antagonist with IC50 of ～6 μM and a selective PPAR-gamma modulator. | ||||
| TN1475 | Caulophyllogenin | 52936-64-8 | 98% |
|
| Caulophyllogenin is a partial PPARγ agonist (EC50 = 12.6 μM) derived from the stem bark of Kalopanax pictus (Araliaceae). Caulophyllogenin inhibits pro-inflammat... | ||||
| TN1804 | Isosilybin A | 142796-21-2 | 98% |
|
| Isosilybin A is a partial PPARγ agonist, it significantly induced ABCA1 protein expression, it inhibited both monophenolase (IC50=1.7-7.6μM) and diphenolase (IC5... | ||||
| T8780 | AMG131 | 315224-26-1 | 98% |
|
| INT-131, is a novel, non-thiazolidinedione (TZD), selective peroxisome proliferator-activated receptor (PPAR)gamma modulator, which can be used for the treatment... | ||||
| T3941 | Choline Fenofibrate | 856676-23-8 | 98% |
|
| Choline Fenofibrate is a choline formulation of fenofibrate, a synthetic phenoxy-isobutyric acid derivate and prodrug with antihyperlipidemic activity. | ||||
| T9808 | Tetradecylthioacetic acid | 2921-20-2 | 98% |
|
| Tetradecylthioacetic acid is a synthetic fatty acid with a sulfur substitution in the β-position. This modification renders TTA unable to undergo complete β-oxid... | ||||
| T1622 | Rosiglitazone maleate | 155141-29-0 | 98% |
|
| Rosiglitazone Maleate is the maleate salt of rosiglitazone, an orally-active thiazolidinedione with antidiabetic properties and potential antineoplastic activity... | ||||
| T77612 | WAY-620472 | 686769-90-4 | 98% |
|
| WAY-620472 is a PPAR regulator that can be used to alter the lifespan of eukaryotes. | ||||
| T9766 | GW590735 | 343321-96-0 | 98% |
|
| GW590735 is an effective and selective PPARα agonist with an EC50 of 4 nM on PPARα and at least 500-fold selectivity versus PPARδ and PPARγ. GW590735 can be used... | ||||
| T1402 | Fenofibric acid | 42017-89-0 | 98% |
|
| Fenofibric Acid is the active form of fenofibrate, a synthetic phenoxy-isobutyric acid derivate with antihyperlipidemic activity. | ||||
| T10900 | CUDA | 479413-68-8 | 98% |
|
| CUDA is an effective soluble cyclohydrolase inhibitor with IC50 of 11.1 nM and 112 nM for mouse sEH and human sEH, respectively. CUDA selectively increases the a... | ||||
| TN4583 | Moringin | 73255-40-0 | 98% |
|
| Moringin is an isothiocyanate obtained from myrosinase-mediated hydrolysis of the glucosinolate precursor glucoMoringin present in Moringa oleifera seeds. Moring... | ||||
| T39516 | Bocidelpar | 2095128-20-2 | 98% |
|
| Bocidelpar is a modulator of PPARδ with an EC50 of 7.80 nM and improves mitochondrial biogenesis and function in Duchenne Muscular Dystrophy muscle cells. | ||||
| T3954 | Adelmidrol | 1675-66-7 | 98% |
|
| Adelmidrol is an anti-inflammatory ethanolamide derivative of azelaic acid. | ||||
| T3056 | Bavachinin | 19879-30-2 | 98% |
|
| Bavachinin(7-O-Methylbavachin) is a natural compound isolated from the Chinese herb Fructus Psoraleae with potent anti-angiogenic activity. | ||||
| T21598L | G3335 Acetate | T21598L | 98% |
|
| G3335 Acetate was discovered to be a novel PPARgamma antagonist. | ||||
| TN1055 | Licochalcone E | 864232-34-8 | 98% |
|
| Licochalcone E is a potential LXRβ agonist. | ||||
| T7159 | L-165041 | 79558-09-1 | 98% |
|
| L-165041 is a potent and selective agonist of the nuclear receptor PPARβ and PPARδ(Ki = 9 nM, EC50 = ~500 nM ,respectively) | ||||
