ペプチド
抗体
色素試薬
PROTAC
バーチャルスクリーニング
TargetMolキット
Cell Counting Kit-8 (CCK-8)
Inhibitor Cocktails
天然化合物
フェノール類
アルカロイド類
フラボノイド類
阻害剤
血管新生
アポトーシス
オートファジー
細胞周期・チェックポイント
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細胞骨格シグナル
DNA損傷・DNA修復
内分泌・ホルモン
GPCR/Gタンパク質
免疫・炎症
JAK・STATシグナル
| Cat. No. | 製品名 | CAS No. | Purity | Chemical Structure |
|---|---|---|---|---|
| T3407 | Rapastinel | 117928-94-6 | 98% |
|
| Rapastinel (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator. | ||||
| T12406 | PEPA | 141286-78-4 | 98% |
|
| PEPA is an allosteric AMPA receptors modulator; binds to the GluA2o and GluA3o LBDs and can be utilized as an indicator of AMPA receptor heterogeneity. | ||||
| T22542 | 1-Aminocyclobutanecarboxylic acid | 22264-50-2 | 98% |
|
| 1-Aminocyclobutanecarboxylic acid is a NMDA receptor partial agonist. 1-Aminocyclobutanecarboxylic acid act at the glycine site, NR1[1]. | ||||
| T2362 | QNZ46 | 1237744-13-6 | 98% |
|
| QNZ46 is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist. | ||||
| T6871 | L-Glutamic acid monosodium salt | 142-47-2 | 98% |
|
| L-Glutamic acid monosodium salt (Monosodium glutamate) is an activator of mGlu1 receptor. | ||||
| T20571 | Cis-PDA | 46026-75-9 | 98% |
|
| cis-PDA, a general ionotropic receptor antagonist, acts by blocking NMDA, AMPA, and kainate mediated responses. It also acts as a partial NMDA receptor agonist. | ||||
| T10930 | D-AP5 | 79055-68-8 | 98% |
|
| D-AP5 is a NMDA receptor antagonist. | ||||
| T1308 | Orphenadrine hydrochloride | 341-69-5 | 98% |
|
| Orphenadrine hydrochloride is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm. | ||||
| T12187L | Naspm trihydrochloride | 1049731-36-3 | 98% |
|
| Naspm trihydrochloride is a synthetic analogue of Joro spider toxin and is an antagonist of calcium permeable AMPA (CP-AMPA) receptors. | ||||
| T0675 | Topiramate | 97240-79-4 | 98% |
|
| Topiramate is a unique antiseizure medication that is used in the treatment of partial and generalized seizures. Topiramate has been rarely associated with hepat... | ||||
| T1443 | Memantine hydrochloride | 41100-52-1 | 98% |
|
| Memantine hydrochloride is an AMANTADINE derivative that has some dopaminergic effects. Memantine hydrochloride has been proposed as an antiparkinson agent. | ||||
| T6352 | (-)-Dizocilpine maleate | 121917-57-5 | 98% |
|
| MK-801 is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes. | ||||
| T22798 | Gavestinel | 153436-38-5 | 98% |
|
| Gavestinel is a non-competitive NMDA receptor antagonist that is potent, selective and orally active.Gavestinel binds to the glycine site of the NMDA receptor wi... | ||||
| T72662 | NMDAR/TRPM4-IN-2 | 2243506-33-2 | 98% |
|
| NMDAR/TRPM4-IN-2 is a potent interfacial inhibitor of NMDAR/TRPM4 interaction.NMDAR/TRPM4-IN-2 protects against MCAO-induced brain damage and NMDA-induced retina... | ||||
| T1946 | Felbamate | 25451-15-4 | 98% |
|
| Felbamate is an Anti-epileptic Agent. The physiologic effect of felbamate is by means of Decreased Central Nervous System Disorganized Electrical Activity. | ||||
| T16964 | SYM2206 | 173952-44-8 | 98% |
|
| SYM2206 is a low affinity non-competitive AMPA receptor antagonist with an IC50 value of 1.6 μM.SYM2206 exhibits anticancer activity by blocking Nav1.6-mediated ... | ||||
| T6618 | Orphenadrine Citrate | 4682-36-4 | 98% |
|
| Orphenadrine Citrate is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects. | ||||
| T1589 | D-Cycloserine | 68-41-7 | 98% |
|
| Cycloserine is a broad spectrum antibiotic used as a second line agent for treatment of drug resistant tuberculosis, always in combination with other antitubercu... | ||||
| T16451 | PEAQX tetrasodium hydrate | T16451 | 98% |
|
| PEAQX tetrasodium hydrate is an orally available NMDA antagonist that is potent and selective. The IC50 value of PEAQX tetrasodium hydrate (459836-30-7 free base... | ||||
| T5819 | Rapastinel Trifluoroacetate | 1435786-04-1 | 98% |
|
| Rapastinel Trifluoroacetate is an NMDA receptor modulator with glycine-site partial agonist properties. | ||||
