Powder: -20°C for 3 years | In solvent: -80°C for 1 year
5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 106,500 |
5 mg | 在庫あり | ¥ 245,500 |
10 mg | 在庫あり | ¥ 328,500 |
25 mg | 在庫あり | ¥ 489,000 |
50 mg | 在庫あり | ¥ 663,500 |
100 mg | 在庫あり | ¥ 890,500 |
ターゲット&IC50 | 5-HT2C receptor:4000 nM, D2 receptor:40 nM, α1-adrenoceptor:10 nM, 5-HT1B receptor:300 nM, 5-HT2A receptor:500 nM, SPLA2:2 nM |
別名 | 5-HT1Amodulator1 |
分子量 | 383.51 |
分子式 | C21H25N3O2S |
CAS No. | 142477-34-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 5 mg/mL (13.04 mM)
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
5-HT1A modulator 1 142477-34-7 GPCR/G Protein Metabolism Neuroscience 5-HT Receptor Dopamine Receptor Phospholipase Adrenergic Receptor 5-HT1Amodulator1 Inhibitor inhibitor inhibit