Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Bay K 8644 (SQ 28,873) is a potent, selective activator of L-type Ca2+ channel with IC50 of 17.3 nM.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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1 mg | 在庫あり | ¥ 8,000 | |||
2 mg | 在庫あり | ¥ 11,000 | |||
5 mg | 在庫あり | ¥ 18,500 | |||
10 mg | 在庫あり | ¥ 29,500 | |||
25 mg | 在庫あり | ¥ 60,500 | |||
50 mg | 在庫あり | ¥ 95,500 | |||
100 mg | 在庫あり | ¥ 142,000 |
説明 | Bay K 8644 (SQ 28,873) is a potent, selective activator of L-type Ca2+ channel with IC50 of 17.3 nM. |
ターゲット&IC50 | Ca2+ channel, L-type:17.3nM(EC50) |
In vitro | Bay K 8644 increases resting tension in segments of mesenteric arteries isolated from young and old rats as an agonist of L-type Ca2+ channel[2] |
In vivo | Bay K 8644 induces small contractions in aortae from Wistar-Kyoto(WKY) rats of 5-week-, 3-month-, 1-year-, 1.5-year-old, which are unaltered with age.[3] |
別名 | (±)-BAY-K-8644, SQ 28,873 |
分子量 | 356.3 |
分子式 | C16H15F3N2O4 |
CAS No. | 71145-03-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ethanol: 35.6 mg/mL (100 mM)
You can also refer to dose conversion for different animals. 詳細
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Bay K 8644 71145-03-4 Membrane transporter/Ion channel Metabolism Calcium Channel (±)-BAY-K-8644 BAY-K 8644 BAY-K8644 influx L-type inhibit sarcolemmal Ca2+ channels Bay K-8644 (±)-Bay K 8644 Inhibitor Bay K8644 BAY-K-8644 SQ 28,873 Ca channels Ca2+ inhibitor