Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CH7057288 is an effective and selective TRK inhibitor with an IC50 value of 1.1 nM, 7.8 nM and 5.1 nM for TRKA, TRKB and TRKC, respectively.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 12,000 | |||
5 mg | 在庫あり | ¥ 28,000 | |||
10 mg | 在庫あり | ¥ 45,500 | |||
25 mg | 在庫あり | ¥ 85,500 | |||
50 mg | 在庫あり | ¥ 128,000 | |||
100 mg | 在庫あり | ¥ 180,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 35,500 |
説明 | CH7057288 is an effective and selective TRK inhibitor with an IC50 value of 1.1 nM, 7.8 nM and 5.1 nM for TRKA, TRKB and TRKC, respectively. |
ターゲット&IC50 | TrkA:1.1 nM , TrkB:7.8 nM , TrkC:5.1 nM |
In vitro | CH7057288, a potent and selective TRK inhibitor belonging to a novel chemical class.CH7057288 induced regression of intracranial tumors and greatly improved event-free survival in an intracranial implantation model mimicking brain metastasis. |
分子量 | 569.67 |
分子式 | C32H31N3O5S |
CAS No. | 2095616-82-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 34 mg/mL (59.68 mM)
You can also refer to dose conversion for different animals. 詳細
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CH7057288 2095616-82-1 Tyrosine Kinase/Adaptors Trk receptor CH-7057288 Inhibitor Trk Receptor inhibit CH 7057288 Tropomyosin related kinase receptor inhibitor