Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Diphylline (Diprophylline) is a xanthine derivative. Diphylline exerts bronchodilator effects and to a lesser extent vasodilator and diuretic properties. Diphylline probably acts as a competitive inhibitor of phosphodiesterase which leads to an increase in intracellular cAMP. This results in relaxation of bronchial smooth muscle and other smooth muscles. Diphylline may also antagonize adenosinereceptors. Diphylline is used in the treatment of acute bronchial asthma, chronic bronchitis and emphysema.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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50 mg | 在庫あり | ¥ 10,000 | |||
100 mg | 在庫あり | ¥ 14,500 | |||
500 mg | 在庫あり | ¥ 41,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 16,000 |
説明 | Diphylline (Diprophylline) is a xanthine derivative. Diphylline exerts bronchodilator effects and to a lesser extent vasodilator and diuretic properties. Diphylline probably acts as a competitive inhibitor of phosphodiesterase which leads to an increase in intracellular cAMP. This results in relaxation of bronchial smooth muscle and other smooth muscles. Diphylline may also antagonize adenosinereceptors. Diphylline is used in the treatment of acute bronchial asthma, chronic bronchitis and emphysema. |
植物由来 |
別名 | Dyphylline, Diprophylline |
分子量 | 254.24 |
分子式 | C10H14N4O4 |
CAS No. | 479-18-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 55 mg/mL (216.33 mM)
H2O: 47 mg/mL (184.9 mM)
Ethanol: < 1 mg/mL (insoluble or slightly soluble)
You can also refer to dose conversion for different animals. 詳細
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Diphylline 479-18-5 GPCR/G Protein Metabolism Neuroscience Adenosine Receptor PDE P1 receptor Dyphylline inhibit Diprophylline Phosphodiesterase (PDE) Inhibitor inhibitor