Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM).
説明 | Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM). |
ターゲット&IC50 | Edg2 receptor:<0.1 μM |
In vitro | Edg-2 receptor inhibitor 1 is an inhibitor of the endothelial differentiation gene receptor 2 (Edg-2, EDG2), which is activated by lysophosphatidic acid (LPA) and is also termed as LPA1 receptor, and is useful for the treatment of diseases such as atherosclerosis, myocardial infarction and heart failure, for example[1]. |
別名 | SAR-100842 |
分子量 | 445.51 |
分子式 | C27H27NO5 |
CAS No. | 1195941-38-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 83.3 mg/mL (186.98 mM)
You can also refer to dose conversion for different animals. 詳細
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Edg-2 receptor inhibitor 1 1195941-38-8 GPCR/G Protein LPA Receptor Edg 2 receptor inhibitor 1 SAR 100842 Edg2 receptor inhibitor 1 SAR100842 SAR-100842 Inhibitor inhibitor inhibit