Powder: -20°C for 3 years | In solvent: -80°C for 1 year
H-9 dihydrochloride is a potent protein kinase (PKA) inhibitor.H-9 Dihydrochloride significantly reduces the excitatory response to 5-HT at low concentrations.H-9 Dihydrochloride affects pharyngeal activity.H-9 Dihydrochloride inhibits signaling and cell growth of EGF ( H-9 Dihydrochloride inhibits EGF (epidermal growth factor)-dependent signaling and cell growth in epithelial cell lines.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 15,000 | |||
5 mg | 在庫あり | ¥ 34,000 | |||
10 mg | 在庫あり | ¥ 51,500 | |||
25 mg | 在庫あり | ¥ 114,500 | |||
50 mg | 在庫あり | ¥ 221,000 | |||
100 mg | 在庫あり | ¥ 296,000 |
説明 | H-9 dihydrochloride is a potent protein kinase (PKA) inhibitor.H-9 Dihydrochloride significantly reduces the excitatory response to 5-HT at low concentrations.H-9 Dihydrochloride affects pharyngeal activity.H-9 Dihydrochloride inhibits signaling and cell growth of EGF ( H-9 Dihydrochloride inhibits EGF (epidermal growth factor)-dependent signaling and cell growth in epithelial cell lines. |
In vitro | Significantly inhibiting A431 cells, H-9 Dihydrochloride is more effective at inhibiting cyclic nucleotide-dependent protein kinases than other kinases[1]. |
In vivo | Microperfusing H-9 Dihydrochloride (100 μM) prevents picrotoxin seizures in 50% of the animals and significantly reduces the mean number of seizures and mean seizure duration[2]. |
分子量 | 324.23 |
分子式 | C11H15Cl2N3O2S |
CAS No. | 116700-36-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: Soluble
You can also refer to dose conversion for different animals. 詳細
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H-9 dihydrochloride 116700-36-8 Angiogenesis GPCR/G Protein JAK/STAT signaling Neuroscience Tyrosine Kinase/Adaptors 5-HT Receptor PKA EGFR H-9 H9 Dihydrochloride H 9 Dihydrochloride H 9 H-9 Dihydrochloride H9 H9 dihydrochloride H 9 dihydrochloride Inhibitor inhibitor inhibit