Powder: -20°C for 3 years | In solvent: -80°C for 1 year
LP-922761 is a potent, selective, and orally active AAK1 inhibitor with inhibitory effects on BMP-2 induced protein kinase (BIKE).
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
2 mg | 在庫あり | ¥ 17,500 | |||
5 mg | 在庫あり | ¥ 30,000 | |||
10 mg | 在庫あり | ¥ 49,000 | |||
25 mg | 在庫あり | ¥ 88,000 | |||
50 mg | 在庫あり | ¥ 130,500 | |||
100 mg | 在庫あり | ¥ 186,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 33,000 |
説明 | LP-922761 is a potent, selective, and orally active AAK1 inhibitor with inhibitory effects on BMP-2 induced protein kinase (BIKE). |
ターゲット&IC50 | AAK1:7.6 nM (cell assays), BIKE:24 nM, AAK1:4.8 nM (enzyme assays) |
In vivo | In mice, the brain-to-plasma ratio of LP-922761 was 0.007, indicating that LP-922761 was basically confined to the peripheral compartment[1]. |
分子量 | 410.47 |
分子式 | C21H26N6O3 |
CAS No. | 1454808-95-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 30 mg/mL (73.09 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
LP-922761 1454808-95-7 Neuroscience AAK1 (AP2 associated kinase 1) LP 922761 LP922761 Inhibitor inhibitor inhibit