Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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サンプルについてお問い合わせ | |||||
5 mg | 在庫あり | ¥ 10,000 | |||
10 mg | 在庫あり | ¥ 13,500 | |||
25 mg | 在庫あり | ¥ 21,000 | |||
50 mg | 在庫あり | ¥ 28,500 | |||
100 mg | 在庫あり | ¥ 36,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 10,500 |
説明 | Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist. |
In vitro | Mequitazine is widely studied and used for allergic disorders such as hay fever and urticaria[1]. Mequitazine demonstrates significant bactericidal effects against all the tested clinical isolates including Ps. aeruginosa. Its effect against the Gram-positive isolates is more pronounced [2]. |
In vivo | Mequitazine antagonizes the effect of histamine in guinea-pig ileum competitively. Mequitazine at 107 produces a parallel shift of the dose-response curve to acetylcholine in the rat duodenum. Mequitazine at highest concentration shows anticholinergic activity [3]. Mequitazine inhibits contractile responses to KCl, phenylephrine (PE), 5-hydroxytryptamine (5-HT), and Ca2+ in rat aorta [4]. |
別名 | Metaplexan, Virginan, Primalan, LM-209 |
分子量 | 322.47 |
分子式 | C20H22N2S |
CAS No. | 29216-28-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (155.05 mM)
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Mequitazine 29216-28-2 GPCR/G Protein Immunology/Inflammation Neuroscience Histamine Receptor LM209 Metaplexan Virginan LM 209 Primalan Inhibitor LM-209 inhibit inhibitor